SCHEMBL6684415

SCHEMBL6684415

COc1ccc(CC(=O)NCc2cn(-c3ccccc3)nc2-c2cccs2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.54
MAPK1 P28482 2/20 0.54
TSHR P16473 1/20 0.54
NPC1 O15118 2/20 0.51
ADORA3 P0DMS8 2/20 0.49
RAB9A P51151 2/20 0.49
POLB P06746 1/20 0.49
KDM4E B2RXH2 4/20 0.48
ALDH1A1 P00352 2/20 0.48
CCNE1 P24864 4/20 0.48
CDK2 P24941 4/20 0.48
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
MEN1 O00255 3/20 0.46
MAPT P10636 3/20 0.46
KMT2A Q03164 3/20 0.46
PPARG P37231 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
NR2E3 Q9Y5X4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6683533 0.91 KDM4E (0.50) SMN1; SMN2MAPK1ADORA3RAB9AKDM4E
SCHEMBL6678678 0.87 ADORA3 (0.60) SMN1; SMN2ADORA3KDM4EALDH1A1CCNE1
SCHEMBL6681136 0.86 MEN1 (0.57) MAPK1ADORA3KDM4EALDH1A1CCNE1
SCHEMBL6677923 0.84 CCNE1 (0.53) SMN1; SMN2MAPK1NPC1ADORA3RAB9A
SCHEMBL6684117 0.81 ALDH1A1 (0.69) SMN1; SMN2MAPK1ADORA3KDM4EALDH1A1
SCHEMBL6677031 0.81 LMNA (0.59) SMN1; SMN2MAPK1TSHRNPC1ADORA3
SCHEMBL6681047 0.80 MEN1 (0.55) MAPK1ADORA3KDM4EALDH1A1MEN1
SCHEMBL6679128 0.79 ALDH1A1 (0.53) SMN1; SMN2ADORA3RAB9APOLBKDM4E
SCHEMBL6679006 0.79 ALDH1A1 (0.56) SMN1; SMN2MAPK1RAB9APOLBKDM4E
SCHEMBL6683539 0.79 ADORA3 (0.54) SMN1; SMN2TSHRNPC1ADORA3RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043951-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS CAREX S.A. (FR) 2004-05-27 WO claimed
WO-2004043951-A1 PYRAZOLE DERIVATIVES AS MODULATORS OF PEROXISOME PROLIFERATOR ACTIVATED RECEPTORS CAREX S.A. (FR) 2004-05-27 WO disclosed