SCHEMBL6684739

SCHEMBL6684739

C1=Nc2ccccc2SCC1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.38
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
RYR2 Q92736 1/20 0.33
HPGD P15428 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29854261 0.78 TRPA1 (0.41) TRPA1
SCHEMBL8276 0.78 TRPA1 (0.41) TRPA1
Hydrochloric Acid SCHEMBL10718555 0.77 TRPA1 (0.39) TRPA1MEN1ALDH1A1GAAKMT2A
SCHEMBL449119 0.70 POLB (0.38) TRPA1MEN1ALDH1A1GAAKMT2A
SCHEMBL28613397 0.68 TRPA1 (0.33) TRPA1
SCHEMBL2516584 0.67 MEN1 (0.34) TRPA1MEN1ALDH1A1GAAKMT2A
SCHEMBL2516583 0.67 TRPA1 (0.38) TRPA1
SCHEMBL1238031 0.67 ALDH1A1 (0.40) TRPA1MEN1ALDH1A1GAAKMT2A
SCHEMBL31001736 0.66 ALDH1A1 (0.48) MEN1ALDH1A1GAAKMT2ARYR2
SCHEMBL255970 0.66 ALDH1A1 (0.48) MEN1ALDH1A1GAAKMT2ARYR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1029847-C Process for preparing 1, 5-benzothiazepine * derivatives TANABE SEIYAKU CO (JP) 1995-09-27 CN claimed
CN-1054597-A Preparation 1, the method for 5-benzothiazepine derivatives TANABE SEIYAKU CO (JP) 1991-09-18 CN claimed
CN-119698413-A Bicyclic tetrahydrothiazepine derivatives 豪夫迈·罗氏有限公司 2025-03-25 CN disclosed
CN-115518402-B Toluene chlorination liquid post-treatment device and treatment method 中盐常州化工股份有限公司 2024-05-28 CN disclosed
CN-116964048-A Bicyclic tetrahydroazepine derivatives for the treatment of cancer 豪夫迈·罗氏有限公司 2023-10-27 CN disclosed
CN-113896612-B Method for selectively preparing o-chlorotoluene 常州新东化工发展有限公司 2023-07-21 CN disclosed
CN-115518402-A Toluene chlorination liquid post-treatment device and treatment method 中盐常州化工股份有限公司 2022-12-27 CN disclosed
CN-101735211-B Applications of 2,3-dihydro[1,5] benzothiazepine compounds or salts thereof in preparation of GSK-3beta inhibitor UNIV FUDAN 2012-11-14 CN disclosed
CN-101735211-B Applications of 2,3-dihydro[1,5] benzothiazepine compounds or salts thereof in preparation of GSK-3beta inhibitor UNIV FUDAN 2012-11-14 CN disclosed
CN-101735211-A 2, application of 3-dihydro [1,5] benzothiaze compounds or salts thereof in preparing GSK-3 beta inhibitor UNIV FUDAN 2010-06-16 CN disclosed
CN-1896078-A Bicyclic pyrrolyl amides as glucogen phosphorylase inhibitors ASTRAZENECA AB (SE) 2007-01-17 CN disclosed
EP-0638082-A1 MACROCYCLIC IMMUNOMODULATORS ABBOTT LABORATORIES (US) 1995-02-15 EP disclosed
WO-1994021642-A1 MACROCYCLIC AMIDE AND UREA IMMUNOMODULATORS ABBOTT LABORATORIES (US) 1994-09-29 WO disclosed
EP-0642516-A4 MACROCYCLIC IMMUNOMODULATORS. ABBOTT LAB (US) 1994-06-15 EP disclosed
EP-0638082-A4 MACROCYCLIC IMMUNOMODULATORS. ABBOTT LAB (US) 1994-06-09 EP disclosed
WO-1993004680-A1 MACROCYCLIC IMMUNOMODULATORS ABBOTT LABORATORIES (US) 1993-03-18 WO disclosed
WO-1993004679-A1 MACROCYCLIC IMMUNOMODULATORS ABBOTT LABORATORIES (US) 1993-03-18 WO disclosed
CN-1005150-B 1, 5-benzothiazepine * derivatives as platelet aggregation inhibitors 田道制药株式会社 1989-09-13 CN disclosed
CN-85101892-A Process for preparing novel 1, 5-benzothiazepine derivatives 1987-01-17 CN disclosed
CN-85103395-A Preparation of 1, 5-benzothiazepine * derivatives as platelet aggregation inhibitors 1986-12-10 CN disclosed