SCHEMBL6684887

SCHEMBL6684887

N#CC(C#N)=Cc1ccc([N+](=O)[O-])cc1O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.56
MAPT P10636 7/20 0.52
ALDH1A1 P00352 6/20 0.52
KDM4E B2RXH2 5/20 0.52
HPGD P15428 3/20 0.52
RECQL P46063 2/20 0.52
LMNA P02545 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
CYP1A2 P05177 1/20 0.52
POLB P06746 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
BLM P54132 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ERN1 O75460 1/20 0.49
GPR35 Q9HC97 2/20 0.49
ERBB2 P04626 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21865015 0.84 EGFR (0.60) EGFRMAPTALDH1A1KDM4EHPGD
SCHEMBL6686433 0.83 MAPT (0.56) EGFRMAPTALDH1A1KDM4EHPGD
SCHEMBL9876993 0.81 MAPT (0.68) EGFRMAPTALDH1A1KDM4EHPGD
SCHEMBL23413367 0.78 ERN1 (0.49) EGFRMAPTALDH1A1HPGDPOLB
SCHEMBL29853796 0.78 ERN1 (0.49) EGFRMAPTALDH1A1HPGDPOLB
SCHEMBL29780565 0.78 ERN1 (0.49) EGFRMAPTALDH1A1HPGDPOLB
SCHEMBL918368 0.76 ERN1 (0.73) MAPTALDH1A1HPGDPOLBERN1
SCHEMBL1353698 0.75 MAPT (0.64) EGFRMAPTALDH1A1KDM4EHPGD
SCHEMBL20302595 0.75 GPR35 (0.56) MAPTALDH1A1KDM4EHPGDPOLB
SCHEMBL3246996 0.75 APP (0.56) EGFRMAPTALDH1A1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487841-A1 THIOPYRIMIDINE AND ISOTHIAZOLOPYRIMIDINE KINASE INHIBITORS Abbott Laboratories (US) 2004-12-22 EP disclosed
WO-2003080625-A1 THIOPYRIMIDINE AND ISOTHIAZOLOPYRIMIDINE KINASE INHIBITORS ABBOTT LABORATORIES (US) 2003-10-02 WO disclosed