SCHEMBL6685745

SCHEMBL6685745

COC(=O)CC(=O)Cc1cc(F)ccc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.43
MAPT P10636 2/20 0.41
HTT P42858 2/20 0.41
RIPK1 Q13546 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.39
SIGMAR1 Q99720 1/20 0.39
ANO1 Q5XXA6 1/20 0.38
MMP2 P08253 2/20 0.38
MMP12 P39900 2/20 0.38
MMP1 P03956 1/20 0.38
MMP9 P14780 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
GPR119 Q8TDV5 1/20 0.38
DPP4 P27487 1/20 0.38
DPP8 Q6V1X1 1/20 0.38
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8063678 0.88 MAPK8 (0.46) MAPK8MAPTHTTRIPK1MEN1
SCHEMBL15778100 0.87 IDO1 (0.46) MAPK8RIPK1SMN1; SMN2ALDH1A1SIGMAR1
SCHEMBL5567382 0.86 MAPT (0.42) MAPK8MAPTHTTRIPK1MEN1
SCHEMBL15778913 0.83 P2RX7 (0.42) MAPTHTTKMT2ASMN1; SMN2ALDH1A1
SCHEMBL6858298 0.82 CES2 (0.48) MAPK8MAPTRIPK1SMN1; SMN2SIGMAR1
SCHEMBL725284 0.81 DPP4 (0.41) MEN1KMT2ASMN1; SMN2ALDH1A1MMP2
SCHEMBL30167907 0.81 DPP4 (0.41) MEN1KMT2ASMN1; SMN2ALDH1A1MMP2
SCHEMBL30434988 0.80 PDGFRB (0.46) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL21061557 0.80 PDGFRB (0.46) MAPTMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL13061970 0.80 RIPK1 (0.49) MAPK8MAPTRIPK1SMN1; SMN2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087650-A2 PROCESS AND INTERMEDIATES FOR THE PREPARATION OF BETA-AMINO ACID AMIDE DIPEPTIDYL PEPTIDASE-IV INHIBITORS MERCK & CO. INC. (US) 2004-10-14 WO disclosed