SCHEMBL6686489

SCHEMBL6686489

NC(=O)c1nc(-c2cccc(Cl)c2)co1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.55
IKBKB O14920 2/20 0.50
RAB9A P51151 3/20 0.48
NPC1 O15118 2/20 0.48
KMO O15229 2/20 0.46
CHUK O15111 1/20 0.45
PARP1 P09874 2/20 0.44
ATP4A P20648 2/20 0.44
ATP4B P51164 2/20 0.44
CNR2 P34972 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ABL1 P00519 1/20 0.42
NOTUM Q6P988 1/20 0.41
JAK2 O60674 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
SLC9A1 P19634 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14564373 0.84 SCN9A (0.62) SCN9AIKBKBKMOPARP1
SCHEMBL8119163 0.81 SCN9A (0.55) SCN9AIKBKBPARP1
SCHEMBL8123493 0.78 SCN9A (0.51) SCN9ARAB9ANPC1SMN1; SMN2
SCHEMBL8153130 0.76 CA2 (0.55) SCN9AIKBKBCHUK
SCHEMBL9955528 0.76 CYP19A1 (0.46) RAB9ANPC1KMOATP4AATP4B
SCHEMBL12170948 0.73 NPC1 (0.66) IKBKBRAB9ANPC1KMOCNR2
SCHEMBL10263341 0.73 ENPP3 (0.59) SCN9ARAB9ANPC1NOTUM
SCHEMBL3821262 0.72 NPC1 (0.59) IKBKBRAB9ANPC1PARP1NOTUM
SCHEMBL5459832 0.72 SCN9A (1.00) SCN9A
SCHEMBL14564400 0.72 SCN9A (0.73) SCN9ARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1442041-A1 AZABICYCLIC-SUBSTITUTED-HETEROARYL COMPOUNDS FOR THE TREATMENT OF DISEASE PHARMACIA & UPJOHN COMPANY (US) 2004-08-04 EP claimed
WO-2003040147-A1 AZABICYCLIC-SUBSTITUTED-HETEROARYL COMPOUNDS FOR THE TREATMENT OF DISEASE__________________________________________________________________________________________________________________________ PHARMACIA & UPJOHN COMPANY (US) 2003-05-15 WO claimed