SCHEMBL9955528

SCHEMBL9955528

Clc1cccc(-c2coc(Cl)n2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.46
NOTUM Q6P988 2/20 0.46
IDO1 P14902 2/20 0.46
ATP4A P20648 2/20 0.44
ATP4B P51164 2/20 0.44
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
RAB9A P51151 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KMO O15229 1/20 0.43
ABL1 P00519 1/20 0.42
MAP4K4 O95819 1/20 0.42
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10263341 0.82 ENPP3 (0.59) NOTUMIDO1NPC1RAB9A
SCHEMBL9954331 0.82 KDM4E (0.50) NOTUMIDO1TP53KMOMAP4K4
SCHEMBL9954530 0.82 ENPP3 (0.59) IDO1ATP4AATP4BNPC1TSHR
SCHEMBL3635042 0.80 MEN1 (0.48) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL3632196 0.78 CYP19A1 (0.48) CYP19A1NOTUMATP4AATP4BNPC1
SCHEMBL14637364 0.76 RAB9A (0.40) NOTUMNPC1RAB9AKMOKDM4E
SCHEMBL3636890 0.76 LTA4H (0.54) CYP19A1NOTUMNPC1TP53RAB9A
SCHEMBL6686489 0.76 SCN9A (0.55) NOTUMATP4AATP4BNPC1RAB9A
SCHEMBL4257536 0.76 HSD17B1 (0.48) NOTUMNPC1TP53TSHRNFKB1
SCHEMBL29470230 0.76 IDO1 (0.55) CYP19A1NOTUMIDO1ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085857-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-3-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed
WO-2012085852-A1 3,8-DIAZA-BICYCLO[4.2.0]OCT-8-YL AMIDES ACTELION PHARMACEUTICALS LTD (CH) 2012-06-28 WO disclosed