SCHEMBL6687217

SCHEMBL6687217

CN(CCNc1cccc(C(N)=O)c1)C(=O)[CH]CC(C)(C)C(N)=O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.42
HTR7 P34969 1/20 0.41
PARP10 Q53GL7 8/20 0.39
PARP14 Q460N5 5/20 0.39
SYK P43405 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC8 Q9BY41 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PARP15 Q460N3 4/20 0.37
GRK2 P25098 1/20 0.37
GRK5 P34947 1/20 0.37
GRK3 P35626 1/20 0.37
DPP4 P27487 1/20 0.36
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.34
ROCK2 O75116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6688710 0.76 POLB (0.43) HDAC1HDAC8HDAC6MEN1KMT2A
SCHEMBL4797902 0.74 PARP1 (0.41) PARP1HTR7PARP10PARP14HDAC1
SCHEMBL18893559 0.70 MEN1 (0.54) PARP1HTR7PARP10PARP14MEN1
SCHEMBL19710767 0.68 HTR7 (0.55) PARP1HTR7PARP10PARP14HDAC8
SCHEMBL8804295 0.67 PARP1 (0.48) PARP1HTR7PARP10PARP14HDAC1
SCHEMBL8294937 0.67 MEN1 (0.57) PARP1PARP10PARP14MEN1KMT2A
SCHEMBL9448456 0.67 PARP1 (0.51) PARP1HTR7PARP10PARP14MEN1
SCHEMBL461708 0.67 HTR7 (0.54) PARP1HTR7PARP10PARP14HDAC8
SCHEMBL21555689 0.66 PARP1 (0.48) PARP1HTR7PARP10PARP14HDAC1
SCHEMBL6688042 0.66 HTR7 (0.39) PARP1HTR7PARP10PARP14MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed