SCHEMBL6688710

SCHEMBL6688710

CN(CCNc1ccc(OC(F)(F)F)cc1)C(=O)[CH]CC(C)(C)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
EPHX2 P34913 1/20 0.39
TDP1 Q9NUW8 3/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
MCHR1 Q99705 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686636 0.89 MAPT (0.42) TDP1KMT2AMEN1MAPTHTT
SCHEMBL6687560 0.86 MAPT (0.38) POLBKMT2AMEN1MAPTHTT
SCHEMBL6689081 0.81 TOP2B (0.36) CA12CA1CA2
SCHEMBL6687217 0.76 PARP1 (0.42) HDAC1HDAC8HDAC6KMT2AMEN1
SCHEMBL6688714 0.76 POLB (0.47) POLBEPHX2TDP1HDAC1HDAC3
SCHEMBL4798680 0.75 CTSS (0.48) POLB
SCHEMBL5500899 0.69 EPHX1 (0.52) POLBHDAC1HDAC3HDAC4HDAC7
SCHEMBL3021858 0.69 EPHX2 (0.57) POLBEPHX2KMT2AMEN1MAPT
SCHEMBL9780251 0.69 EPHX2 (0.56) POLBEPHX2TDP1HDAC1HDAC3
SCHEMBL6685718 0.69 TDP1 (0.48) POLBEPHX2TDP1L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084843-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed