SCHEMBL6687243

SCHEMBL6687243

COc1ccc(NCCNC(=O)C(CCNC(=O)c2ccc(C#N)cc2)C2CCCCC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.53
CTSL P07711 12/20 0.53
CTSK P43235 8/20 0.51
MAPT P10636 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MDM2 Q00987 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6689172 0.85 CTSS (0.61) CTSSCTSLCTSK
SCHEMBL6691132 0.83 CTSS (0.69) CTSSCTSLCTSKMAPTRAB9A
SCHEMBL6685381 0.82 CTSL (0.75) CTSSCTSLCTSK
SCHEMBL6685236 0.82 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL6691086 0.81 CTSS (0.59) CTSSCTSLCTSK
SCHEMBL5842763 0.81 CTSS (0.72) CTSSCTSLCTSK
SCHEMBL5842769 0.81 CTSS (0.72) CTSSCTSLCTSK
SCHEMBL6687973 0.81 EPHX2 (0.50) CTSSCTSLCTSKNPC1RAB9A
SCHEMBL5843852 0.81 CTSS (0.78) CTSSCTSLCTSK
SCHEMBL5843860 0.81 CTSS (0.78) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084842-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed