SCHEMBL6691132

SCHEMBL6691132

COc1ccc(NCCNC(=O)C(CCNC(=O)c2ccc(N3CCOCC3)cc2)C2CCCCC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.69
CTSL P07711 9/20 0.69
CTSK P43235 7/20 0.69
RAB9A P51151 2/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NR4A1 P22736 1/20 0.47
KMT2A Q03164 1/20 0.47
MCL1 Q07820 1/20 0.47
TP53 P04637 1/20 0.46
POLB P06746 1/20 0.46
LCK P06239 1/20 0.45
JAK3 P52333 1/20 0.45
GFER P55789 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687243 0.83 CTSS (0.53) CTSSCTSLCTSKRAB9AMAPT
SCHEMBL5843384 0.82 CTSS (0.85) CTSSCTSLCTSK
SCHEMBL5843387 0.82 CTSS (0.85) CTSSCTSLCTSK
SCHEMBL6689172 0.81 CTSS (0.61) CTSSCTSLCTSK
SCHEMBL6685381 0.80 CTSL (0.75) CTSSCTSLCTSK
SCHEMBL6692650 0.78 CTSS (0.60) CTSSCTSLCTSK
SCHEMBL6691086 0.77 CTSS (0.59) CTSSCTSLCTSK
SCHEMBL6693346 0.77 CTSS (0.69) CTSSCTSLCTSK
SCHEMBL6690368 0.75 CTSS (0.58) CTSSCTSLCTSKALDH1A1KMT2A
SCHEMBL6690169 0.75 CTSL (0.73) CTSSCTSLCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004084842-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-10-07 WO disclosed