SCHEMBL6687470

SCHEMBL6687470

COc1cc(CN[C@@H](Cc2ccccc2)C(N)=O)ccc1OCc1ccc(OC(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSD P07339 2/20 0.56
NPC1 O15118 1/20 0.49
PKM P14618 1/20 0.49
RAB9A P51151 1/20 0.49
MRGPRX1 Q96LB2 2/20 0.48
F2 P00734 1/20 0.48
F10 P00742 1/20 0.48
PRSS1 P07477 1/20 0.48
F7 P08709 1/20 0.48
BCHE P06276 1/20 0.46
MTNR1A P48039 2/20 0.46
MTNR1B P49286 2/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2C19 P33261 1/20 0.45
CAPN1 P07384 1/20 0.45
PPARG P37231 1/20 0.44
ALDH1A1 P00352 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687466 1.00 CTSD (0.56) CTSDNPC1PKMRAB9AMRGPRX1
SCHEMBL6686899 0.90 NPC1 (0.58) NPC1PKMRAB9AMRGPRX1F2
SCHEMBL6686902 0.90 NPC1 (0.58) NPC1PKMRAB9AMRGPRX1F2
SCHEMBL6686193 0.89 CTSD (0.55) CTSDNPC1PKMRAB9AMRGPRX1
SCHEMBL6686196 0.89 CTSD (0.55) CTSDNPC1PKMRAB9AMRGPRX1
SCHEMBL6685490 0.87 ATM (0.48) CTSDNPC1PKMRAB9AMRGPRX1
SCHEMBL6685493 0.87 ATM (0.48) CTSDNPC1PKMRAB9AMRGPRX1
SCHEMBL6687236 0.85 MAOB (0.51) CTSDNPC1PKMRAB9A
SCHEMBL6687232 0.85 MAOB (0.51) CTSDNPC1PKMRAB9A
SCHEMBL6693520 0.85 MTNR1A (0.55) CTSDNPC1PKMRAB9AMRGPRX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed