SCHEMBL668763

SCHEMBL668763

O=C(O)n1ccc2cc(C(F)(F)F)ccc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.43
PIM2 Q9P1W9 1/20 0.43
CES2 O00748 2/20 0.42
S1PR1 P21453 1/20 0.42
CCR2 P41597 1/20 0.40
KRAS P01116 1/20 0.40
PPARD Q03181 3/20 0.40
PPARA Q07869 3/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
OXER1 Q8TDS5 1/20 0.38
PPARG P37231 1/20 0.38
IDH1 O75874 1/20 0.38
KDR P35968 1/20 0.38
PKM P14618 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL668802 0.84 OXER1 (0.35) S1PR1KRASPPARDPPARAOXER1
SCHEMBL28682739 0.83 KCNH2 (0.41) PIM1PIM2CES2S1PR1KRAS
SCHEMBL31517105 0.83 KCNH2 (0.41) PIM1PIM2CES2S1PR1KRAS
SCHEMBL20905231 0.81 KRAS (0.53) PIM1PIM2S1PR1KRASMEN1
SCHEMBL15218078 0.79 MAP2K4 (0.45) KRASIDH1KDRKCNH2
SCHEMBL17674406 0.77 TFPI2 (0.55) CCR2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2651525 0.76 PIM1 (0.47) PIM1PPARDPPARAKDM4EKMT2A
SCHEMBL16619618 0.75 CA2 (0.52) PIM1PIM2CES2CCR2KRAS
SCHEMBL4959132 0.74 PRKCI (0.52) CCR2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2659180 0.74 OXER1 (0.63) PIM1CCR2OXER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9758453-B2 One-component reagent for the fluoroalkylation reaction THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2017-09-12 US disclosed
US-20170066717-A1 NEW PHENYLAZETIDINECARBOXYLATE OR -CARBOXAMIDE COMPOUNDS INVENTIVA (FR) 2017-03-09 US disclosed
US-20160185691-A1 One-Component Reagent for the Fluoroalkylation Reaction THE BOARD OF TRUSTEES OF THE UNIVERSITY OF LLLINOIS (US) 2016-06-30 US disclosed
US-9193648-B2 Fluoroalkylation methods and reagents BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2015-11-24 US disclosed
US-20130225815-A1 Fluoroalkylation Methods And Reagents THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2013-08-29 US disclosed
EP-2606048-A1 FLUOROALKYLATION METHODS AND REAGENTS The Board of Trustees of the University of Illinois (US) 2013-06-26 EP disclosed
WO-2012024564-A1 FLUOROALKYLATION METHODS AND REAGENTS THE BOARD OF TRUSTESS OF THE UNIVERSITY OF ILLINOIS (US) 2012-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130225815-A1 Fluoroalkylation Methods And Reagents ALK, AFF4, AFF2 PIM1 1415/4885PIM2 1176/4885CES2 744/4885
US-20170066717-A1 NEW PHENYLAZETIDINECARBOXYLATE OR -CARBOXAMIDE COMPOUNDS NCOR1, NCOR2, NCOA1 PIM1 1594/4885PIM2 2416/4885CES2 2319/4885
US-20160185691-A1 One-Component Reagent for the Fluoroalkylation Reaction AOC1, AOC3, AOC2 PIM1 4530/4885PIM2 4612/4885CES2 98/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.