SCHEMBL6687908

SCHEMBL6687908

COc1cc(CNC(C)C(N)=O)ccc1OCc1c(F)cccc1F

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.56
MEN1 O00255 2/20 0.56
SCN9A Q15858 2/20 0.53
MAOB P27338 6/20 0.53
MAOA P21397 4/20 0.53
SMN1; SMN2 Q16637 1/20 0.49
GAA P10253 1/20 0.48
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687911 1.00 KMT2A (0.56) KMT2AMEN1SCN9AMAOBMAOA
SCHEMBL6686469 0.89 KMT2A (0.53) KMT2AMEN1SCN9AMAOBMAOA
SCHEMBL6686470 0.89 KMT2A (0.53) KMT2AMEN1SCN9AMAOBMAOA
SCHEMBL6690744 0.86 KMT2A (0.53) KMT2AMEN1SMN1; SMN2GAAALDH1A1
SCHEMBL6685320 0.86 KMT2A (0.55) KMT2AMEN1SMN1; SMN2GAAALDH1A1
SCHEMBL6690750 0.86 KMT2A (0.53) KMT2AMEN1SMN1; SMN2GAAALDH1A1
SCHEMBL6690285 0.86 KMT2A (0.55) KMT2AMEN1SMN1; SMN2GAAALDH1A1
SCHEMBL8802147 0.84 ALDH1A1 (0.60) KMT2AMEN1SCN9AMAOBMAOA
SCHEMBL2995936 0.83 SCN9A (0.74) KMT2ASCN9AMAOBMAOAGAA
SCHEMBL2995932 0.83 SCN9A (0.74) KMT2ASCN9AMAOBMAOAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed