SCHEMBL6687960

SCHEMBL6687960

COc1cccc(COc2ccc(CN[C@@H](Cc3ccccc3)C(N)=O)cc2)c1

nearest known ligand 0.64

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.56
MAOA P21397 1/20 0.55
SCN9A Q15858 1/20 0.55
BCHE P06276 1/20 0.54
PPARG P37231 1/20 0.52
HDAC8 Q9BY41 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687957 1.00 MAOB (0.56) MAOBMAOASCN9ABCHEPPARG
SCHEMBL6690337 0.95 MAOB (0.54) MAOBMAOASCN9A
SCHEMBL6690341 0.95 MAOB (0.54) MAOBMAOASCN9A
SCHEMBL6693523 0.89 MTNR1A (0.55)
SCHEMBL6693520 0.89 MTNR1A (0.55)
SCHEMBL1070366 0.84 MAOB (0.76) MAOBMAOASCN9A
SCHEMBL6690014 0.84 MTNR1A (0.54) BCHE
SCHEMBL6690026 0.84 MTNR1A (0.54) BCHE
SCHEMBL6687983 0.82 MRGPRX4 (0.50)
SCHEMBL6687988 0.82 MRGPRX4 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO claimed
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed