SCHEMBL6693523

SCHEMBL6693523

COc1cccc(COc2ccc(CN[C@@H](Cc3ccccc3)C(N)=O)cc2OC)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.55
MTNR1B P49286 1/20 0.55
CTSD P07339 6/20 0.54
ABCB1 P08183 1/20 0.53
POLB P06746 2/20 0.51
ALDH1A1 P00352 1/20 0.51
NPC1 O15118 1/20 0.50
PKM P14618 1/20 0.50
RAB9A P51151 1/20 0.50
CAPN1 P07384 1/20 0.49
MRGPRX1 Q96LB2 2/20 0.49
F2 P00734 1/20 0.48
F10 P00742 1/20 0.48
PRSS1 P07477 1/20 0.48
F7 P08709 1/20 0.48
MRGPRX4 Q96LA9 1/20 0.47
CSF1R P07333 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6693520 1.00 MTNR1A (0.55) MTNR1AMTNR1BCTSDABCB1POLB
SCHEMBL6690026 0.95 MTNR1A (0.54) MTNR1AMTNR1BCTSDABCB1POLB
SCHEMBL6690014 0.95 MTNR1A (0.54) MTNR1AMTNR1BCTSDABCB1POLB
SCHEMBL6686902 0.92 NPC1 (0.58) MTNR1AMTNR1BALDH1A1NPC1PKM
SCHEMBL6686899 0.92 NPC1 (0.58) MTNR1AMTNR1BALDH1A1NPC1PKM
SCHEMBL6687960 0.89 MAOB (0.56)
SCHEMBL6687957 0.89 MAOB (0.56)
SCHEMBL6693045 0.85 MTNR1A (0.52) MTNR1AMTNR1BCTSDABCB1POLB
SCHEMBL6687983 0.85 MRGPRX4 (0.50) MTNR1AMTNR1BNPC1RAB9AMRGPRX4
SCHEMBL6693042 0.85 MTNR1A (0.52) MTNR1AMTNR1BCTSDABCB1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed