SCHEMBL6687983

SCHEMBL6687983

COc1cccc(COc2ccc(CNC(Cc3ccc(O)cc3)C(N)=O)cc2Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 2/20 0.50
CD274 Q9NZQ7 5/20 0.44
MTNR1A P48039 2/20 0.43
MTNR1B P49286 1/20 0.43
FFAR1 O14842 1/20 0.43
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
XBP1 P17861 1/20 0.42
HTT P42858 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
ANO1 Q5XXA6 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6687988 1.00 MRGPRX4 (0.50) MRGPRX4CD274MTNR1AMTNR1BFFAR1
SCHEMBL6690014 0.90 MTNR1A (0.54) MTNR1AMTNR1BNPC1RAB9A
SCHEMBL6690026 0.90 MTNR1A (0.54) MTNR1AMTNR1BNPC1RAB9A
SCHEMBL6690337 0.87 MAOB (0.54)
SCHEMBL6690341 0.87 MAOB (0.54)
SCHEMBL6693520 0.85 MTNR1A (0.55) MRGPRX4MTNR1AMTNR1BNPC1RAB9A
SCHEMBL6693523 0.85 MTNR1A (0.55) MRGPRX4MTNR1AMTNR1BNPC1RAB9A
SCHEMBL6687960 0.82 MAOB (0.56)
SCHEMBL6687957 0.82 MAOB (0.56)
SCHEMBL6690108 0.77 SMN1; SMN2 (0.56) MAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087125-A1 AMINO ACID DERIVATIVES AS INHIBITORS OF MAMMALIAN SODIUM CHANNELS IONIX PHARMACEUTICALS LIMITED (GB) 2004-10-14 WO disclosed