SCHEMBL6688939

SCHEMBL6688939

Cc1ccc(OCNC2CC2)cc1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.58
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
DRD2 P14416 3/20 0.43
DRD4 P21917 3/20 0.43
DRD3 P35462 3/20 0.43
ALDH1A1 P00352 1/20 0.41
WDR5 P61964 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2474020 0.85 KDM4E (0.60) KDM4ECYP1A2CYP2D6CYP2C19MEN1
SCHEMBL2467576 0.81 KDM4E (0.79) KDM4ECYP1A2CYP2D6CYP2C19MEN1
SCHEMBL5562491 0.81 ATF4 (0.54) KDM4E
SCHEMBL2471205 0.80 KMT2A (0.50) KDM4EMEN1KMT2ADRD2DRD4
SCHEMBL1824874 0.80 MEN1 (0.43) MEN1KMT2ADRD2DRD4DRD3
SCHEMBL2473347 0.79 KMT2A (0.48) KDM4EMEN1KMT2ADRD2DRD4
SCHEMBL13980799 0.75 KDM4E (0.68) KDM4ECYP1A2CYP2D6CYP2C19MEN1
SCHEMBL23074658 0.74 KDM4E (0.88) KDM4ECYP1A2CYP2D6CYP2C19MEN1
SCHEMBL23074654 0.74 KDM4E (0.88) KDM4ECYP1A2CYP2D6CYP2C19MEN1
SCHEMBL14097162 0.73 DRD2 (0.50) KDM4EDRD2DRD4DRD3WDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004105762-A1 MEDICAL USE OF DIAZABICYCLONONENE DERIVATIVES AS INHIBITORS OF PARASITE ASPARTIC PROTEASES ACTELION PHARMACEUTICALS LTD (CH) 2004-12-09 WO disclosed