SCHEMBL6689303

SCHEMBL6689303

CCCCC(C(=O)c1nc2ccccc2o1)(C(NC1CCCCC1)C(N)=O)S(=O)(=O)CC1CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FAAH O00519 4/20 0.36
CTSS P25774 6/20 0.36
XDH P47989 1/20 0.35
CES1 P23141 1/20 0.35
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
MAPT P10636 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6632064 0.77 FAAH (0.37) FAAHCTSSXDHCES1NPC1
SCHEMBL6685143 0.68 CTSS (0.46) CTSS
SCHEMBL6650333 0.68 CTSS (0.46) CTSS
SCHEMBL6061887 0.68 CTSS (0.46) CTSS
SCHEMBL6062621 0.68 CTSS (0.46) CTSS
SCHEMBL6695509 0.66 FAAH (0.40) FAAHCTSSXDHCES1MAPT
SCHEMBL6467110 0.66 CTSS (0.44) FAAHCTSSCES1NPC1RAB9A
SCHEMBL6062624 0.66 FAAH (0.42) FAAHCTSSCES1LMNASMN1; SMN2
SCHEMBL6061894 0.66 FAAH (0.42) FAAHCTSSCES1LMNASMN1; SMN2
SCHEMBL6651561 0.63 NPC1 (0.33) NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP disclosed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO disclosed