SCHEMBL6651561

SCHEMBL6651561

CCCCC(c1cccs1)(C(NC1CCOCC1)C(N)=O)C(O)c1nc2ccccc2o1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
POLB P06746 1/20 0.32
PTPN2 P17706 1/20 0.31
PTPN1 P18031 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6651565 0.75 TSHR (0.38) NPC1RAB9APOLBPTPN2PTPN1
SCHEMBL6062924 0.68 REN (0.37) NPC1RAB9A
SCHEMBL6062927 0.68 REN (0.37) NPC1RAB9A
SCHEMBL6062920 0.68 REN (0.37) NPC1RAB9A
SCHEMBL6629735 0.66 FOLH1 (0.37) NPC1RAB9A
SCHEMBL6696965 0.65 TP53 (0.34)
SCHEMBL6687639 0.65 CTSK (0.38) NPC1RAB9APTPN2PTPN1
SCHEMBL6685881 0.64 PTPN1 (0.40) NPC1RAB9APTPN2PTPN1
SCHEMBL6689303 0.63 FAAH (0.36) NPC1RAB9A
SCHEMBL6652838 0.62 CTSS (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397340-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2004-03-17 EP disclosed
WO-2002098850-A2 CHEMICAL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-12-12 WO disclosed