SCHEMBL6690440

SCHEMBL6690440

CS(=O)(=O)c1ccc(CNC(=O)c2ccncc2C#CC(Cl)c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 12/20 0.46
CYP2C9 P11712 3/20 0.46
CCR1 P32246 3/20 0.42
MAPK8 P45983 1/20 0.41
MAPK9 P45984 1/20 0.41
MAPK10 P53779 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6238040 0.79 NAMPT (0.51) NAMPTCYP2C9CCR1MAPK8MAPK9
SCHEMBL6232551 0.79 NAMPT (0.50) NAMPTCYP2C9MAPK8MAPK9MAPK10
SCHEMBL6233999 0.72 NAMPT (0.46) NAMPTCYP2C9CCR1MAPK8MAPK9
SCHEMBL16088664 0.69 APEX1 (0.74) CCR1TSHRHSD17B10CYP2C19ALDH1A1
SCHEMBL933885 0.68 TSHR (0.67) NAMPTCYP2C9TSHRHSD17B10ALDH1A1
SCHEMBL933289 0.68 EPHX2 (0.68) NAMPTCYP2C9TDP1HSD17B10ALDH1A1
SCHEMBL933464 0.67 ALDH1A1 (0.72) TSHRHSD17B10ALDH1A1
SCHEMBL5814687 0.67 KMT2A (0.76) MAPK8MAPK9MAPK10HSD17B10ALDH1A1
SCHEMBL1053062 0.67 ALDH1A1 (0.53) NAMPTCYP2C9CCR1HSD17B10ALDH1A1
SCHEMBL6266349 0.67 NR1H4 (0.42) NAMPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1434585-A1 ALKYNE MATRIX METALLOPROTEINASE INHIBITORS Warner-Lambert Company LLC (US) 2004-07-07 EP claimed
WO-2003032999-A1 ALKYNE MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2003-04-24 WO claimed