SCHEMBL933289

SCHEMBL933289

CS(=O)(=O)c1ccc(CNC(=O)c2ccncc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.68
NR1H4 Q96RI1 1/20 0.68
CA2 P00918 2/20 0.66
L3MBTL1 Q9Y468 1/20 0.64
LMNA P02545 2/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
TDP1 Q9NUW8 1/20 0.58
NAMPT P43490 3/20 0.58
CYP2C9 P11712 1/20 0.58
CA1 P00915 1/20 0.57
GAA P10253 2/20 0.55
ROCK2 O75116 1/20 0.54
RPS6KA5 O75582 1/20 0.54
MAP4K4 O95819 1/20 0.54
PRKCG P05129 1/20 0.54
PRKACA P17612 1/20 0.54
RPS6KB1 P23443 1/20 0.54
MAPK1 P28482 1/20 0.54
AKT1 P31749 1/20 0.54
GSK3A P49840 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23199278 0.94 CA2 (0.74) EPHX2NR1H4CA2LMNASMN1; SMN2
SCHEMBL933464 0.85 ALDH1A1 (0.72) EPHX2NR1H4CA2LMNACA1
SCHEMBL13658737 0.84 NR1H4 (0.74) EPHX2NR1H4CA2CA1GAA
SCHEMBL933885 0.83 TSHR (0.67) EPHX2NR1H4CA2LMNANAMPT
SCHEMBL12810429 0.82 EPHX2 (0.72) EPHX2NR1H4CA2L3MBTL1LMNA
SCHEMBL1569157 0.82 L3MBTL1 (0.77) CA2L3MBTL1LMNASMN1; SMN2GAA
SCHEMBL1568232 0.81 SMN1; SMN2 (0.74) L3MBTL1LMNASMN1; SMN2TDP1NAMPT
SCHEMBL8374098 0.81 L3MBTL1 (0.71) CA2L3MBTL1LMNASMN1; SMN2CYP2C9
SCHEMBL19358856 0.81 ALDH1A1 (0.76) CA2LMNASMN1; SMN2TDP1NAMPT
SCHEMBL22059471 0.81 EPHX2 (1.00) EPHX2NR1H4CA2L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed