SCHEMBL933464

SCHEMBL933464

CS(=O)(=O)c1ccc(CNC(=O)c2ccccc2)cc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.72
GAA P10253 1/20 0.72
HSD17B10 Q99714 1/20 0.72
EPHX2 P34913 1/20 0.72
NR1H4 Q96RI1 1/20 0.72
KDM4E B2RXH2 1/20 0.67
POLB P06746 1/20 0.67
TSHR P16473 1/20 0.67
RECQL P46063 1/20 0.67
CA2 P00918 3/20 0.64
HDAC1 Q13547 4/20 0.63
HDAC6 Q9UBN7 3/20 0.63
CA1 P00915 2/20 0.62
LMNA P02545 1/20 0.59
RORC P51449 1/20 0.59
HDAC3 O15379 2/20 0.58
ADAMTS4 O75173 1/20 0.58
CA12 O43570 1/20 0.58
CA9 Q16790 1/20 0.58
HDAC2 Q92769 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13658737 0.89 NR1H4 (0.74) ALDH1A1GAAHSD17B10EPHX2NR1H4
SCHEMBL29488705 0.86 RORC (0.71) ALDH1A1KDM4EPOLBTSHRRECQL
SCHEMBL933289 0.85 EPHX2 (0.68) ALDH1A1GAAHSD17B10EPHX2NR1H4
SCHEMBL12810429 0.85 EPHX2 (0.72) EPHX2NR1H4KDM4EPOLBTSHR
SCHEMBL5681681 0.85 HDAC1 (0.64) ALDH1A1GAAHSD17B10EPHX2KDM4E
SCHEMBL5677882 0.84 CA2 (0.88) EPHX2NR1H4CA2CA1CA12
SCHEMBL16088664 0.84 APEX1 (0.74) ALDH1A1GAAHSD17B10EPHX2NR1H4
SCHEMBL22059471 0.84 EPHX2 (1.00) EPHX2NR1H4CA2HDAC6CA1
SCHEMBL933885 0.83 TSHR (0.67) ALDH1A1GAAHSD17B10EPHX2NR1H4
SCHEMBL28266792 0.83 RORC (0.83) ALDH1A1GAAHSD17B10EPHX2NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114436955-A Tetrahydroquinoline and benzomorpholine derivatives or salts thereof, and preparation method and application thereof 复旦大学 2022-05-06 CN disclosed
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed