SCHEMBL6691852

SCHEMBL6691852

O=c1ccccn1-c1cc(-c2nc3cc(C(F)(F)F)ccc3s2)cc(-c2ccccc2Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGPAT2 O15120 3/20 0.44
ILK Q13418 2/20 0.39
MAT2A P31153 1/20 0.36
AKR1B1 P15121 4/20 0.36
AKR1B10 O60218 1/20 0.36
AKR1A1 P14550 1/20 0.36
GLO1 Q04760 1/20 0.36
HSD11B1 P28845 1/20 0.36
DYRK1A Q13627 1/20 0.35
PDE2A O00408 1/20 0.35
PDE10A Q9Y233 1/20 0.35
KDM4E B2RXH2 2/20 0.34
S1PR2 O95136 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1884283 0.78 AGPAT2 (0.44) AGPAT2ILKAKR1B1AKR1B10AKR1A1
SCHEMBL2138665 0.70 ILK (0.54) AGPAT2ILKDYRK1AKDM4EALDH1A1
SCHEMBL6691854 0.70 AGPAT2 (0.46) AGPAT2ILKMAT2AAKR1B1AKR1B10
SCHEMBL12470403 0.66 ILK (0.56) AGPAT2ILKDYRK1AKDM4EALDH1A1
SCHEMBL29348201 0.66 CYP2A6 (0.48) POLB
SCHEMBL7259223 0.66 AGPAT2 (0.60) AGPAT2ILKDYRK1AKDM4EALDH1A1
SCHEMBL12470914 0.66 ILK (0.52) AGPAT2ILKDYRK1AKDM4EALDH1A1
SCHEMBL11011940 0.65 ILK (0.52) AGPAT2ILKAKR1B1AKR1B10AKR1A1
SCHEMBL1885251 0.65 GRIA1 (0.51) AGPAT2ILKAKR1B1AKR1B10AKR1A1
SCHEMBL8704110 0.65 KDM4E (0.55) AGPAT2ILKDYRK1AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed