SCHEMBL6693024

SCHEMBL6693024

CC(C)(C)OC(=O)NC[C@@H](CS(C)(=O)=O)C1CNc2ccc(F)cc21

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.36
EPHX2 P34913 1/20 0.34
CCNT1 O60563 3/20 0.33
CDK9 P50750 3/20 0.33
HTR1A P08908 1/20 0.33
HTR1D P28221 1/20 0.33
HTR1F P30939 1/20 0.33
RORC P51449 2/20 0.33
F12 P00748 6/20 0.32
PCSK9 Q8NBP7 1/20 0.32
F2 P00734 2/20 0.32
ACACB O00763 1/20 0.32
CTSS P25774 1/20 0.32
CTSK P43235 1/20 0.32
AAK1 Q2M2I8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4973253 0.81 CTSS (0.42) GPR119EPHX2CCNT1CDK9CTSS
SCHEMBL6686186 0.74 CCNT1 (0.36) EPHX2CCNT1CDK9RORC
SCHEMBL6694455 0.74 CTSS (0.39) GPR119EPHX2CCNT1CDK9PCSK9
SCHEMBL6690191 0.73 F12 (0.40) F12F2
SCHEMBL2258801 0.65 KMT2A (0.39) HTR1AHTR1DHTR1FF12
SCHEMBL6687211 0.64 F12 (0.38) HTR1AHTR1DHTR1FF12F2
SCHEMBL29135644 0.63 MKNK2 (0.44) GPR119AAK1
SCHEMBL6689109 0.63 MEN1 (0.41) CTSSCTSKAAK1
SCHEMBL2375918 0.62 MKNK2 (0.45) EPHX2CTSSCTSKAAK1
SCHEMBL5484730 0.62 HTR1A (0.44) GPR119CCNT1CDK9HTR1AHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004112709-A2 INHIBITORS OF CATHEPSIN S IRM LLC (BM) 2004-12-29 WO disclosed