SCHEMBL6693260

SCHEMBL6693260

N#Cc1ccccc1-c1ccccc1-c1cc(-c2cscn2)c[nH]c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.42
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
PIK3CD O00329 1/20 0.40
PIK3CA P42336 1/20 0.40
PIK3CB P42338 1/20 0.40
GRIA1 P42261 1/20 0.39
GRIA3 P42263 1/20 0.39
PDE4D Q08499 1/20 0.39
IDO1 P14902 2/20 0.39
TDO2 P48775 1/20 0.39
CDK2 P24941 1/20 0.38
GSK3B P49841 1/20 0.38
SCN9A Q15858 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36
MAPK1 P28482 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15758398 0.82 GRIA1 (0.57) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL687843 0.81 GRIA1 (0.58) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL6695727 0.79 MCL1 (0.47) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL6693263 0.77 MCL1 (0.40) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL1536988 0.75 MAPK1 (0.47) KDM4EIDO1TDO2SCN9AMAPK1
SCHEMBL1887741 0.74 GRIA1 (0.71) KDM4EALDH1A1GRIA1GRIA3PDE4D
SCHEMBL18007259 0.73 MCL1 (0.49) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL20267848 0.66 MCL1 (0.41) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL10707443 0.65 MCL1 (0.63) MCL1KDM4EALDH1A1HPGDPIK3CD
SCHEMBL4082911 0.65 MAPK1 (0.41) IDO1TDO2SCN9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed