SCHEMBL6695727

SCHEMBL6695727

N#Cc1ccccc1-c1ccccc1-c1cc(-c2ncccn2)c[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.47
KDM4E B2RXH2 4/20 0.47
HPGD P15428 3/20 0.47
ALDH1A1 P00352 2/20 0.47
PIK3CD O00329 1/20 0.45
PIK3CA P42336 1/20 0.45
PIK3CB P42338 1/20 0.45
PDE4D Q08499 2/20 0.45
GRIA1 P42261 1/20 0.45
GRIA3 P42263 1/20 0.45
TNKS O95271 5/20 0.43
TNKS2 Q9H2K2 1/20 0.43
PRMT5 O14744 1/20 0.39
WDR77 Q9BQA1 1/20 0.39
GALR3 O60755 1/20 0.38
GAA P10253 1/20 0.38
USP8 P40818 1/20 0.38
USP7 Q93009 1/20 0.38
CLK4 Q9HAZ1 1/20 0.37
PDE5A O76074 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15758398 0.87 GRIA1 (0.57) MCL1KDM4EHPGDALDH1A1PIK3CD
SCHEMBL687843 0.86 GRIA1 (0.58) MCL1KDM4EHPGDALDH1A1PIK3CD
SCHEMBL18007259 0.83 MCL1 (0.49) MCL1KDM4EHPGDALDH1A1PIK3CD
SCHEMBL6693260 0.79 MCL1 (0.42) MCL1KDM4EHPGDALDH1A1PIK3CD
SCHEMBL6692469 0.78 TNKS (0.44) TNKSTNKS2
SCHEMBL6695728 0.74 MCL1 (0.45) MCL1KDM4EHPGDALDH1A1PIK3CD
SCHEMBL6131063 0.71 ESR2 (0.47) HPGDALDH1A1PDE4DGRIA1GRIA3
SCHEMBL1882537 0.71 GRIA1 (0.79) KDM4EALDH1A1PDE4DGRIA1GRIA3
SCHEMBL16456315 0.71 TNKS (0.52) KDM4ETNKSTNKS2GAALMNA
SCHEMBL10707443 0.70 MCL1 (0.63) MCL1KDM4EHPGDALDH1A1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465626-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES Eisai Co., Ltd. (JP) 2004-10-13 EP disclosed
WO-2003047577-A2 PHARMACEUTICAL COMPOSITIONS COMPRISING DIHYDROPYRIDINONE COMPOUNDS AND AN IMMUNOREGULATORY OR AN ANTIINFLAMMATORY AGENT AND THEIR USES EISAI CO LTD (JP) 2003-06-12 WO disclosed