SCHEMBL669373

SCHEMBL669373

CCC(OS(C)(=O)=O)(c1cccc(OC)c1)C(C)CN(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.38
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
HTR2A P28223 2/20 0.38
MRGPRX2 Q96LB1 1/20 0.38
CHRM3 P20309 1/20 0.38
HRH2 P25021 1/20 0.38
ADRA1A P35348 1/20 0.38
OPRK1 P41145 1/20 0.38
CYP2D6 P10635 3/20 0.38
CYP3A4 P08684 2/20 0.38
LMNA P02545 1/20 0.38
ALDH1A1 P00352 2/20 0.35
CYP2C19 P33261 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
AOC3 Q16853 2/20 0.34
PER2 O15055 1/20 0.33
CRY1 Q16526 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL669655 1.00 KCNH2 (0.38) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL14974361 1.00 KCNH2 (0.38) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL14984858 1.00 KCNH2 (0.38) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL14987837 0.91 HTR2A (0.37) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL17750791 0.85 CYP2D6 (0.40) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL22454446 0.85 CYP2D6 (0.40) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL669770 0.85 LMNA (0.39) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL669526 0.85 LMNA (0.39) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL14974352 0.85 LMNA (0.39) KCNH2OPRM1OPRD1HTR2AMRGPRX2
SCHEMBL14987836 0.82 KCNH2 (0.41) KCNH2OPRM1OPRD1HTR2AMRGPRX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606030-A1 PROCESS FOR THE PREPARATION OF TAPENTADOL Indoco Remedies Limited (IN) 2013-06-26 EP disclosed
WO-2012023147-A1 PROCESS FOR THE PREPARATION OF TAPENTADOL INDOCO REMEDIES LIMITED (IN) 2012-02-23 WO disclosed