SCHEMBL6694965

SCHEMBL6694965

Cc1ccc2c(Nc3ccc4[nH]ncc4c3)nc(-c3cccnc3)nc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.60
MAPK1 P28482 2/20 0.60
HTT P42858 1/20 0.60
TGFBR1 P36897 1/20 0.55
ROCK2 O75116 6/20 0.54
ABCG2 Q9UNQ0 7/20 0.52
ABCB1 P08183 2/20 0.52
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
TSHR P16473 2/20 0.51
CLK4 Q9HAZ1 2/20 0.51
USP2 O75604 1/20 0.51
ALDH1A1 P00352 1/20 0.51
LMNA P02545 1/20 0.51
KDM4E B2RXH2 2/20 0.51
HPGD P15428 1/20 0.51
CYP2C19 P33261 1/20 0.51
HSD17B10 Q99714 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
KDM1A O60341 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL3581668 0.91 ROCK2 (0.55) MAPTMAPK1HTTTGFBR1ROCK2
SCHEMBL6694913 0.89 LATS1 (0.57) MAPTTGFBR1ROCK2ABCG2ABCB1
SCHEMBL6925655 0.88 ROCK2 (0.54) MAPTMAPK1HTTTGFBR1ROCK2
SCHEMBL3581272 0.88 TGFBR1 (0.58) MAPTTGFBR1ROCK2ABCG2ABCB1
SCHEMBL3587684 0.86 TGFBR1 (0.56) MAPTTGFBR1ROCK2ABCG2ABCB1
SCHEMBL3582617 0.85 ROCK2 (0.56) MAPTTGFBR1ROCK2ABCG2ABCB1
SCHEMBL3586795 0.84 TGFBR1 (0.54) MAPTTGFBR1ROCK2ABCG2ABCB1
SCHEMBL3585279 0.82 TNIK (0.54) TGFBR1ROCK2ABCG2ABCB1CLK4
SCHEMBL14475760 0.82 ABCG2 (0.66) ROCK2ABCG2ABCB1CYP1A2CYP3A4
SCHEMBL14474835 0.82 MAPT (0.64) MAPTMAPK1HTTABCG2ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065392-A1 CONDENSED PYRIDINES AND PYRIMIDINES AND THEIR USE AS ALK-5 RECEPTOR LIGANDS SMITHKLINE BEECHAM CORPORATION (US) 2004-08-05 WO disclosed