SCHEMBL6695860

SCHEMBL6695860

C[S+]([O-])c1ccc(-c2oc(-c3ccccc3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.52
MAPK13 O15264 2/20 0.52
MAPK12 P53778 2/20 0.52
MAPK11 Q15759 2/20 0.52
GCGR P47871 1/20 0.52
USP1 O94782 1/20 0.47
USP19 O94966 1/20 0.47
UCHL3 P15374 1/20 0.47
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
HPGD P15428 2/20 0.43
CYP2C19 P33261 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
POLB P06746 1/20 0.43
HSP90AA1 P07900 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
HTT P42858 1/20 0.43
CCR6 P51684 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7503500 1.00 MAPK14 (0.52) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL1387188 0.90 MAPK14 (0.65) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL16993493 0.90 MAPK14 (0.65) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL9113400 0.86 MAPK14 (0.61) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL8549078 0.81 PTGS2 (0.40) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL1387186 0.81 MAPK14 (0.71) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL8553156 0.80 PTGS2 (0.68) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL7504194 0.80 PTGS2 (0.68) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL213979 0.80 PTGS2 (0.68) MAPK14MAPK13MAPK12MAPK11GCGR
SCHEMBL7503429 0.79 MAPK14 (0.81) MAPK14MAPK13MAPK12MAPK11GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096206-A2 THERAPEUTIC COMBINATION OF A COX-2 INHIBITOR AND A TACE INHIBITOR PHARMACIA CORPORATION (US) 2004-11-11 WO disclosed