SCHEMBL8549078

SCHEMBL8549078

C[S+]([O-])c1ccc(-c2oc(C(c3ccccc3)c3ccccc3)nc2-c2ccc(F)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.40
PTGS1 P23219 3/20 0.40
MAPK14 Q16539 4/20 0.38
CYP1A2 P05177 1/20 0.38
POLB P06746 1/20 0.38
HSP90AA1 P07900 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 1/20 0.38
CCR6 P51684 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
MAPK11 Q15759 3/20 0.36
MAPK13 O15264 2/20 0.36
MAPK12 P53778 2/20 0.36
GCGR P47871 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6695860 0.81 MAPK14 (0.52) PTGS2PTGS1MAPK14CYP1A2POLB
SCHEMBL7503500 0.81 MAPK14 (0.52) PTGS2PTGS1MAPK14CYP1A2POLB
SCHEMBL7503544 0.81 PTGS2 (0.64) PTGS2PTGS1
SCHEMBL9024375 0.79 PTGS2 (0.65) PTGS2PTGS1CYP1A2POLBHSP90AA1
SCHEMBL7499074 0.79 PTGS2 (0.62) PTGS2PTGS1PTGDR2
SCHEMBL8295663 0.76 KMT2A (0.39) PTGS2PTGS1CYP1A2POLBHSP90AA1
SCHEMBL1387188 0.74 MAPK14 (0.65) PTGS2PTGS1MAPK14MAPK11MAPK13
SCHEMBL16993493 0.74 MAPK14 (0.65) PTGS2PTGS1MAPK14MAPK11MAPK13
SCHEMBL9025437 0.73 PTGS2 (0.45) PTGS2PTGS1MAPK14CYP3A4HPGD
SCHEMBL8551444 0.71 PTGS2 (0.39) PTGS2PTGS1MAPK14MAPK11MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed