SCHEMBL6698680

SCHEMBL6698680

CC(C)c1ccc(-c2cc(Cl)ccc2C2=NC(C)(C)CO2)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
IL2 P60568 1/20 0.36
ATM Q13315 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HRH3 Q9Y5N1 2/20 0.34
CYP2D6 P10635 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6698687 0.84 HRH3 (0.39) HTTLMNAMAPTKDM4EHRH3
SCHEMBL8560175 0.82 HTT (0.41) HTTLMNAMAPTKDM4EHPGD
SCHEMBL7489373 0.80 KDM4E (0.49) HTTLMNAMAPTKDM4EATM
SCHEMBL11491135 0.78 KDM4E (0.47) HTTLMNAMAPTKDM4EHPGD
SCHEMBL7497195 0.77 KDM4E (0.43) HTTLMNAMAPTKDM4EHPGD
SCHEMBL7831700 0.76 KDM4E (0.45) HTTLMNAMAPTKDM4EHPGD
SCHEMBL9463701 0.76 KDM4E (0.40) HTTLMNAMAPTKDM4EHPGD
SCHEMBL655887 0.75 HPGD (0.46) HTTLMNAMAPTKDM4EHPGD
SCHEMBL3762622 0.74 KDM4E (0.51) HTTLMNAMAPTKDM4EHPGD
SCHEMBL9016431 0.74 KDM4E (0.43) HTTLMNAMAPTKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040044008-A1 Use of therapeutic benzamide derivatives DAUGAN ALAIN CLAUDE-MARIE (FR) 2004-03-04 US disclosed
US-6552022-B1 Atherosclerosis in a mammal, pancreatitis, non-insulin dependent diabetes mellitus, coronary heart disease in a lowering serum lipid levels SMITHKLINE BEECHAM CORPORATION 2003-04-22 US disclosed
EP-1286670-A2 USE OF THERAPEUTIC BENZAMIDE DERIVATIVES GLAXO GROUP LIMITED (GB) 2003-03-05 EP disclosed
WO-2001097810-A2 USE OF THERAPEUTIC BENZAMIDE DERIVATIVES GLAXO GROUP LIMITED (GB) 2001-12-27 WO disclosed
EP-1135378-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2001-09-26 EP disclosed
WO-2000032582-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS APOB-100 SECRETION INHIBITORS GLAXO GROUP LIMITED (GB) 2000-06-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040044008-A1 Use of therapeutic benzamide derivatives MTTP, LIPC, CETP HTT 2382/4885LMNA 1661/4885MAPT 2320/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.