SCHEMBL8560175

SCHEMBL8560175

Cc1ccc(-c2ccc(Cl)cc2C2=NC(C)(C)CO2)cc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.41
LMNA P02545 2/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 2/20 0.40
IL2 P60568 1/20 0.40
HPGD P15428 2/20 0.39
ATM Q13315 2/20 0.37
ALDH1A1 P00352 2/20 0.37
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
CYP2D6 P10635 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6698680 0.82 HTT (0.40) HTTLMNAMAPTKDM4EIL2
SCHEMBL371 0.81 KDM4E (0.49) HTTLMNAMAPTKDM4EIL2
SCHEMBL7831700 0.81 KDM4E (0.45) HTTLMNAMAPTKDM4EIL2
SCHEMBL7934334 0.81 KDM4E (0.45) HTTLMNAMAPTKDM4EIL2
SCHEMBL11491135 0.80 KDM4E (0.47) HTTLMNAMAPTKDM4EIL2
SCHEMBL11080851 0.80 KDM4E (0.42) HTTLMNAMAPTKDM4EIL2
SCHEMBL3942245 0.77 KDM4E (0.53) HTTLMNAMAPTKDM4EIL2
SCHEMBL498998 0.77 KDM4E (0.44) HTTLMNAMAPTKDM4EHPGD
SCHEMBL655887 0.77 HPGD (0.46) HTTLMNAMAPTKDM4EHPGD
SCHEMBL4472084 0.76 HTT (0.52) HTTLMNAMAPTKDM4EIL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0598702-B1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same EISAI CO LTD (JP) 1998-06-10 EP disclosed
EP-0628557-B1 Biphenylmethane derivatives, the use of them and pharmacological compositions containing same EISAI CO LTD (JP) 1997-05-02 EP disclosed
US-5506238-A HYPOTENSIVE AGENT EISAI CO., LTD. (JP) 1996-04-09 US disclosed
EP-0420237-B1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same EISAI CO LTD (JP) 1996-03-06 EP disclosed
EP-0628557-A1 Biphenylmethane derivatives, the use of them and pharmacological compositions containing same Eisai Co., Ltd. (JP) 1994-12-14 EP disclosed
US-5328911-A Cardiovascular disorders, hypotensive agents and congestive heart failure EISAI CO., LTD. (JP) 1994-07-12 US disclosed
EP-0598702-A1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same Eisai Co., Ltd. (JP) 1994-05-25 EP disclosed
US-5298518-A Biphenylmethane derivative and pharmacological use EISAI CO., LTD. (JP) 1994-03-29 US disclosed
EP-0420237-A1 Biphenylmethane derivative, the use of it and pharmacological compositions containing same Eisai Co., Ltd. (JP) 1991-04-03 EP disclosed