SCHEMBL669877

SCHEMBL669877

O=Cc1ccc(-c2ccc(F)cc2F)c(Cl)c1Cl

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.38
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
NFE2L2 Q16236 4/20 0.37
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
PTPN1 P18031 1/20 0.34
DPP4 P27487 1/20 0.34
LMNA P02545 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
DHFR P00374 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
TTR P02766 1/20 0.33
ALB P02768 1/20 0.33
HMGB1 P09429 1/20 0.33
HPGD P15428 1/20 0.33
CXCL12 P48061 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16518103 0.79 ERN1 (0.46) ERN1PIM1PIM3TDP1ALDH1A1
SCHEMBL16616202 0.79 ERN1 (0.40) ERN1PIM1PIM3NFE2L2ALDH1A1
SCHEMBL19154298 0.75 NFE2L2 (0.47) ERN1PIM1PIM3NFE2L2TDP1
SCHEMBL96915 0.75 NFE2L2 (0.54) ERN1NFE2L2ALDH1A1KDM4EPTPN1
SCHEMBL29824365 0.75 NFE2L2 (0.54) ERN1NFE2L2ALDH1A1KDM4EPTPN1
SCHEMBL16616115 0.75 ERN1 (0.49) ERN1PIM1PIM3ALDH1A1KDM4E
SCHEMBL505574 0.74 PIM1 (0.50) ERN1PIM1PIM3NFE2L2ALDH1A1
SCHEMBL6495322 0.73 TDP1 (0.46) ERN1TDP1LMNAMEN1KMT2A
SCHEMBL16616040 0.72 ERN1 (0.42) ERN1ALDH1A1MEN1CA1CA2
SCHEMBL14879562 0.72 ALDH1A1 (0.49) NFE2L2ALDH1A1KDM4ELMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2605658-A1 SPIROXAZOLIDINONE COMPOUNDS Merck Sharp & Dohme Corp. (US) 2013-06-26 EP disclosed
WO-2012024183-A1 SPIROXAZOLIDINONE COMPOUNDS MERCK SHARP & DOHME CORP. (US) 2012-02-23 WO disclosed