SCHEMBL6699643

SCHEMBL6699643

N=C(N)NC(=O)N(F)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 3/20 0.35
CYP3A4 P08684 2/20 0.35
MAPT P10636 2/20 0.35
CYP2C19 P33261 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
CYP1A2 P05177 2/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
PLAU P00749 1/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
BLM P54132 2/20 0.33
F2 P00734 1/20 0.33
F10 P00742 1/20 0.33
F12 P00748 1/20 0.33
F7 P08709 1/20 0.33
F3 P13726 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347561 0.85 NPSR1 (0.39) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
SCHEMBL28899661 0.81 ALDH1A1 (0.36) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
SCHEMBL6695684 0.79 PLAU (0.38) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
SCHEMBL6691760 0.79 NPSR1 (0.36) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
SCHEMBL28515349 0.79 NPSR1 (0.36) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
Bicarbonate SCHEMBL27820467 0.77 NPSR1 (0.41) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
SCHEMBL9518724 0.75 NPSR1 (0.43) NPSR1ALDH1A1TDP1L3MBTL1MEN1
SCHEMBL6694934 0.75 MEN1 (0.59) ALDH1A1L3MBTL1MEN1KMT2AF2
SCHEMBL8396658 0.74 NPSR1 (0.46) NPSR1ALDH1A1CYP3A4MAPTCYP2C19
SCHEMBL5490024 0.73 L3MBTL1 (0.42) NPSR1ALDH1A1CYP3A4CYP2C19TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3553083-B2 2004-08-11 JP claimed
EP-0852494-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-07-15 EP claimed
WO-1997009973-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-03-20 WO claimed