SCHEMBL6701352

SCHEMBL6701352

CC(C)C(O)(CCc1ccc(F)cc1C(F)(F)F)CC(=O)n1ccnc1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 9/20 0.35
THRB P10828 1/20 0.35
SLC6A4 P31645 5/20 0.34
SLC6A2 P23975 4/20 0.34
SLC6A3 Q01959 2/20 0.34
NTRK1 P04629 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CYP3A4 P08684 1/20 0.33
HTR2A P28223 1/20 0.33
DHFR P00374 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6691020 0.87 HTT (0.36) THRBSLC6A4SLC6A2CYP3A4
SCHEMBL6692213 0.82 NR3C2 (0.39) P2RX7THRBCYP3A4
SCHEMBL6699765 0.82 CYP19A1 (0.42)
SCHEMBL6694672 0.81 CYP11B1 (0.42)
SCHEMBL6699772 0.79 HMOX1 (0.41)
SCHEMBL6694121 0.78 CYP24A1 (0.33) THRB
SCHEMBL6693514 0.77 SLC13A5 (0.34)
SCHEMBL6696472 0.77 MEN1 (0.40) HTR2A
SCHEMBL6694813 0.76 CYP24A1 (0.43)
SCHEMBL6694999 0.72 LNPEP (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040106606-A1 HIV protease inhibitors BOYER FREDERICK EARL (US) 2004-06-03 US claimed
US-6528510-B1 Dihydropyrones with tethered heterocycles; 3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsulfanyl)-4-hydroxy-6 -isopropyl-6-(2-pyridin-4-yl-ethyl)-5,6-dihydro-pyran - 2-one; WARNER-LAMBERT COMPANY 2003-03-04 US claimed
EP-1112269-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-07-04 EP claimed
WO-2000015634-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2000-03-23 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040106606-A1 HIV protease inhibitors DNPEP, PREP, PEPD P2RX7 4258/4885THRB 4765/4885SLC6A4 3154/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.