SCHEMBL6696472

SCHEMBL6696472

CC(C)C(O)(CCc1cccc(C(F)(F)F)c1)CC(=O)n1ccnc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
EPHX1 P07099 3/20 0.39
NR3C2 P08235 1/20 0.39
MC4R P32245 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
HTR2B P41595 1/20 0.38
GRM2 Q14416 1/20 0.37
GRM3 Q14832 1/20 0.37
CACNA1G O43497 1/20 0.37
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
TAAR1 Q96RJ0 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
CETP P11597 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6694672 0.88 CYP11B1 (0.42) NR3C2CACNA1GNPC1
SCHEMBL6699772 0.88 HMOX1 (0.41) ALDH1A1
SCHEMBL6692213 0.83 NR3C2 (0.39) EPHX1NR3C2GRM2
SCHEMBL6699765 0.81 CYP19A1 (0.42)
SCHEMBL6691020 0.80 HTT (0.36) MEN1KMT2ANR3C2ALDH1A1LMNA
SCHEMBL6303531 0.79 SLC13A5 (0.51) MEN1KMT2AEPHX1HTR2AHTR2C
SCHEMBL6701352 0.77 P2RX7 (0.35) HTR2A
SCHEMBL6694999 0.77 LNPEP (0.35) GRM2GRM3
SCHEMBL7642170 0.77 HMOX1 (0.52)
SCHEMBL7642166 0.77 HMOX1 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040106606-A1 HIV protease inhibitors BOYER FREDERICK EARL (US) 2004-06-03 US claimed
US-6528510-B1 Dihydropyrones with tethered heterocycles; 3-(2-tert-Butyl-4-hydroxymethyl-5-methyl-phenylsulfanyl)-4-hydroxy-6 -isopropyl-6-(2-pyridin-4-yl-ethyl)-5,6-dihydro-pyran - 2-one; WARNER-LAMBERT COMPANY 2003-03-04 US claimed
EP-1112269-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2001-07-04 EP claimed
WO-2000015634-A2 HIV PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 2000-03-23 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040106606-A1 HIV protease inhibitors DNPEP, PREP, PEPD MEN1 3684/4885KMT2A 2939/4885EPHX1 1267/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.