Cadaverine Tartrate

Cadaverine Tartrate

SCHEMBL6701773

CC(C)COc1ccc(CC(=O)N(Cc2ccc(F)cc2)C2CCN(C3CCOCC3)CC2)cc1.O=C(O)C(O)C(O)C(=O)O

nearest known ligand 0.57

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3CHRM1CHRM2CHRM3CHRM4ESR1ESR2GABRA1GABRB1GABRG2GBA1HRH1HTR1DHTR2AOPRD1OPRK1OPRM1SLC6A2SLC6A3TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8rplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cadaverine Tartrate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 20/20 0.57
ADRB2 known ✓ P07550 1/20 0.53
CHRM2 known ✓ P08172 1/20 0.53
CHRM1 known ✓ P11229 1/20 0.53
SLC6A2 known ✓ P23975 1/20 0.53
ADRA1A known ✓ P35348 1/20 0.53
OPRM1 known ✓ P35372 1/20 0.53
SLC6A3 known ✓ Q01959 1/20 0.53
ABCB11 O95342 1/20 0.53
CYP1A2 P05177 1/20 0.53
DRD1 P21728 1/20 0.53
TBXA2R P21731 1/20 0.53
HTR2C P28335 1/20 0.53
GPR183 P32249 1/20 0.53
CYP2C19 P33261 1/20 0.53
APLNR P35414 1/20 0.53
DRD3 P35462 1/20 0.53
CX3CR1 P49238 1/20 0.53
KCNH2 Q12809 1/20 0.53
GPR65 Q8IYL9 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL339279 0.95 HTR2A (0.61) HTR2AABCB11CYP1A2ADRB2CHRM2
Cadaverine Tartrate SCHEMBL10322724 0.92 HTR2A (0.59) HTR2AABCB11CYP1A2ADRB2CHRM2
Cadaverine Tartrate SCHEMBL10322313 0.90 HTR2A (0.46) HTR2AOPRM1
Cadaverine Tartrate SCHEMBL10321944 0.89 HTR2A (0.55) HTR2AABCB11CYP1A2ADRB2CHRM2
Cadaverine Tartrate SCHEMBL3946014 0.88 HTR2A (0.56) HTR2AABCB11CYP1A2ADRB2CHRM2
SCHEMBL366677 0.87 HTR2A (0.64) HTR2AABCB11CYP1A2ADRB2CHRM2
SCHEMBL20794614 0.85 HTR2A (0.57) HTR2AABCB11CYP1A2ADRB2CHRM2
SCHEMBL20767064 0.85 HTR2A (0.57) HTR2AABCB11CYP1A2ADRB2CHRM2
Cadaverine Tartrate SCHEMBL10322265 0.84 HTR2A (0.56) HTR2AABCB11CYP1A2ADRB2CHRM2
Cadaverine Tartrate SCHEMBL10321720 0.84 HTR2A (0.56) HTR2AABCB11CYP1A2ADRB2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2983473-A2 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS Mountain Llc (US) 2016-02-17 EP claimed
US-20140350064-A1 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS MOUNTAIN LLC 2014-11-27 US claimed
WO-2014144130-A2 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS MOUNTAIN LLC (US) 2014-09-18 WO claimed
EP-2983473-A2 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS Mountain Llc (US) 2016-02-17 EP disclosed
US-20140350064-A1 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS MOUNTAIN LLC 2014-11-27 US disclosed
WO-2014144130-A2 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS MOUNTAIN LLC (US) 2014-09-18 WO disclosed
US-20120183600-A1 NOVEL COMPOSITION FOR TREATING METABOLIC SYNDROME AND OTHER CONDITIONS CHEN CHIEN-HUNG (US) 2012-07-19 US disclosed
US-20040106600-A1 N-substituted piperidine derivatives as serotonin receptor agents ACADIA PHARMACEUTICALS, INC. 2004-06-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040106600-A1 N-substituted piperidine derivatives as serotonin receptor agents HTR1A, HTR5A, HTR1B HTR2A 12/4885ADRB2 158/4885CHRM2 250/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.