SCHEMBL6704579

SCHEMBL6704579

Cc1cccc(-c2nc(Nc3ccc4[nH]ncc4c3)c3cc(Cl)ccc3n2)n1

nearest known ligand 0.79

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 14/20 0.79
PAK4 O96013 2/20 0.51
ROCK2 O75116 4/20 0.48
MAPK14 Q16539 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6684201 0.88 TGFBR1 (1.00) TGFBR1ROCK2MAPK14
SCHEMBL30814808 0.88 TGFBR1 (1.00) TGFBR1ROCK2MAPK14
SCHEMBL3592877 0.83 TGFBR1 (0.54) TGFBR1PAK4ROCK2
SCHEMBL3590264 0.81 PAK4 (0.53) TGFBR1PAK4ROCK2
SCHEMBL3588932 0.80 ROCK2 (0.63) TGFBR1ROCK2
SCHEMBL3578380 0.80 PAK4 (0.52) TGFBR1PAK4ROCK2
SCHEMBL3578657 0.79 TNIK (0.53) TGFBR1PAK4ROCK2
SCHEMBL5736843 0.77 ROCK2 (0.56) TGFBR1PAK4ROCK2MAPK14
SCHEMBL3583464 0.77 ROCK2 (0.58) TGFBR1PAK4ROCK2
Hydrochloric Acid SCHEMBL3581146 0.76 ROCK2 (0.56) TGFBR1PAK4ROCK2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065392-A1 CONDENSED PYRIDINES AND PYRIMIDINES AND THEIR USE AS ALK-5 RECEPTOR LIGANDS SMITHKLINE BEECHAM CORPORATION (US) 2004-08-05 WO disclosed