SCHEMBL670916

SCHEMBL670916

Ic1ccc(Nc2ccccc2)nc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 1/20 0.56
MAPT P10636 4/20 0.53
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
LMNA P02545 1/20 0.53
PDGFRB P09619 3/20 0.47
PDGFRA P16234 3/20 0.47
RAB9A P51151 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
KDM4E B2RXH2 1/20 0.47
ALPG P10696 1/20 0.47
GRM5 P41594 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CDK2 P24941 2/20 0.43
MAPK1 P28482 2/20 0.43
NPC1 O15118 2/20 0.43
CHEK1 O14757 1/20 0.43
IKBKB O14920 1/20 0.43
AURKA O14965 1/20 0.43
PDPK1 O15530 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22938770 0.88 HCAR3 (0.42) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL21666862 0.83 EDNRA (0.36) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL22788044 0.79 RAB9A (0.59) MAPTRAB9AKDM4ECDK2NPC1
SCHEMBL31532396 0.76 ALDH1A1 (0.60) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL913981 0.76 HCAR3 (0.56) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL21258720 0.76 HCAR3 (0.56) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL2280918 0.76 ALDH1A1 (0.60) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL21258996 0.76 HCAR3 (0.56) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL83157 0.76 HCAR3 (0.56) HCAR3MAPTMEN1KMT2ALMNA
SCHEMBL28513546 0.75 RAB9A (0.62) MEN1KMT2ALMNARAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606052-A1 NICOTINIC RECEPTOR COMPOUNDS Research Triangle Institute (US) 2013-06-26 EP disclosed
WO-2012024615-A1 NICOTINIC RECEPTOR COMPOUNDS RESEARCH TRIANGLE INSTITUTE (US) 2012-02-23 WO disclosed
EP-2268143-A2 NOVEL PIPERIDINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE Forest Laboratories Holdings Limited (BM) 2011-01-05 EP disclosed
WO-2009117676-A2 NOVEL PIPERIDINE DERIVATIVES AS INHIBITORS OF STEAROYL-COA DESATURASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2009-09-24 WO disclosed