SCHEMBL671067

SCHEMBL671067

COC(=O)c1cccc(CN2CCNCC2=O)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 2/20 0.53
LOXL2 Q9Y4K0 1/20 0.50
CYP4F2 P78329 2/20 0.49
CYP4A11 Q02928 2/20 0.49
ABHD6 Q9BV23 1/20 0.48
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
MAPK10 P53779 1/20 0.47
GSK3B P49841 1/20 0.46
PARP1 P09874 1/20 0.45
IDO1 P14902 1/20 0.45
MAPT P10636 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
SLC7A5 Q01650 1/20 0.44
MRGPRX4 Q96LA9 1/20 0.44
CD74 P04233 1/20 0.44
MIF P14174 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL670624 0.85 CYP2C9 (0.55) IDO1MAPTL3MBTL1MEN1ALDH1A1
SCHEMBL22346843 0.82 LOXL2 (0.52) LOXL2CYP4F2CYP4A11ABHD6ROCK2
SCHEMBL1512308 0.82 CHRM3 (0.72) CHRM3LOXL2CYP4F2CYP4A11MEN1
SCHEMBL27554554 0.80 PRSS1 (0.47) LOXL2
SCHEMBL671044 0.79 LOXL2 (0.48) LOXL2CYP4F2CYP4A11ABHD6ROCK2
SCHEMBL675320 0.78 LOXL2 (0.50) LOXL2CYP4F2CYP4A11ABHD6ROCK2
SCHEMBL3154100 0.78 POLB (0.67) CHRM3MAPTMEN1ALDH1A1KMT2A
SCHEMBL31773 0.78 LOXL2 (0.52) LOXL2CYP4F2CYP4A11ABHD6ROCK2
Hydrochloric Acid SCHEMBL6417883 0.77 SLC6A2 (0.44) CHRM3MAPTMIFMEN1KMT2A
Trifluoroacetic Acid SCHEMBL1018573 0.75 CHRM3 (0.63) CHRM3LOXL2MEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012024179-A1 SUBSTITUTED AMIDE DERIVATIVES AS DGAT-1 INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-02-23 WO disclosed