SCHEMBL6720856

SCHEMBL6720856

O=C(O)CCc1ccccc1OS(=O)(=O)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.48
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
FFAR4 Q5NUL3 5/20 0.43
KEAP1 Q14145 1/20 0.41
FFAR1 O14842 6/20 0.40
PTGER1 P34995 3/20 0.40
PTGER4 P35408 3/20 0.40
PTGER3 P43115 3/20 0.40
PTGER2 P43116 3/20 0.40
LTB4R Q15722 2/20 0.40
LTB4R2 Q9NPC1 2/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
KMT2A Q03164 1/20 0.40
PTGDR Q13258 1/20 0.39
DHFR P00374 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6938219 0.84 DRD2 (0.38)
SCHEMBL27219471 0.83 CXCL8 (0.48) NPSR1FFAR4MEN1KMT2A
SCHEMBL4376769 0.81 DRD2 (0.46) LTB4RLTB4R2
SCHEMBL3721270 0.80 MAPT (0.49) NPSR1THRATHRBKEAP1FFAR1
SCHEMBL30055829 0.80 FFAR1 (0.56) NPSR1THRATHRBFFAR4KEAP1
SCHEMBL1508357 0.80 FFAR1 (0.56) NPSR1THRATHRBFFAR4KEAP1
SCHEMBL13604212 0.79 DRD2 (0.46) NPSR1
SCHEMBL2829914 0.79 DRD2 (0.44) THRATHRB
SCHEMBL7369905 0.78 POLB (0.53) NPSR1KEAP1FFAR1ALDH1A1
Iodide SCHEMBL9652564 0.78 DRD2 (0.44) THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1478619-A1 A PROCESS FOR PREPARING A PHENYLALANINE DERIVATIVE AND INTERMEDIATES THEREOF TANABE SEIYAKU CO., LTD. (JP) 2004-11-24 EP disclosed
WO-2003072536-A1 A PROCESS FOR PREPARING A PHENYLALANINE DERIVATIVE AND INTERMEDIATES THEREOF TANABE SEIYAKU CO., LTD. (JP) 2003-09-04 WO disclosed
US-5496805-A DIURETIC, HYPOTENSIVE E. R. SQUIBB & SONS, INC. (US) 1996-03-05 US disclosed