SCHEMBL6721147

SCHEMBL6721147

Oc1c(Cl)cc(C#Cc2ccccc2)cc1Cl

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 2/20 0.71
AKR1C1 Q04828 2/20 0.71
APP P05067 1/20 0.52
HNF4A P41235 1/20 0.43
TTR P02766 3/20 0.42
HSD17B10 Q99714 3/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP3A4 P08684 2/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
MAPT P10636 3/20 0.41
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.39
GRM5 P41594 1/20 0.39
FFAR1 O14842 2/20 0.39
FFAR4 Q5NUL3 1/20 0.39
GRM4 Q14833 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18130077 0.77 APP (0.57) AKR1C2AKR1C1APPHNF4AHSD17B10
SCHEMBL717466 0.76 APP (0.55) AKR1C2AKR1C1APPHNF4AMAPT
SCHEMBL2450399 0.75 APP (0.80) AKR1C2AKR1C1APPHNF4AHSD17B10
SCHEMBL4267409 0.75 APP (0.60) AKR1C2AKR1C1APPHNF4AHSD17B10
SCHEMBL20211704 0.75 APP (0.60) AKR1C2AKR1C1APPHNF4AHSD17B10
SCHEMBL18549484 0.74 APP (0.67) AKR1C2AKR1C1APPHNF4AHSD17B10
SCHEMBL717647 0.74 APP (0.67) AKR1C2AKR1C1APPHNF4AHSD17B10
SCHEMBL19026498 0.73 APP (0.57) AKR1C2AKR1C1APPHNF4AMAPT
Diphenylacetylene SCHEMBL960609 0.72 APP (1.00) APPHSD17B10ALDH1A1CYP3A4TSHR
Diphenylacetylene SCHEMBL29188592 0.72 APP (1.00) APPHSD17B10ALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6677473-B1 TREATMENT, PREVENTION OR AMELIORATION OF ONE OR MORE SYMPTOMS OF THROMBOTIC DISORDERS, UNSTABLE ANGINA OR CANCER CORVAS INTERNATIONAL INC 2004-01-13 US disclosed
WO-2001036351-A2 PLASMINOGEN ACTIVATOR INHIBITOR ANTAGONISTS RELATED APPLICATIONS CORVAS INTERNATIONAL, INC. (US) 2001-05-25 WO disclosed