SCHEMBL6724438

SCHEMBL6724438

CN(C)C1(c2cccs2)CCC(NC(Cc2c[nH]c3ccccc23)C(=O)O)CC1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.50
OPRL1 P41146 3/20 0.50
ITGB2 P05107 4/20 0.49
ICAM1 P05362 4/20 0.49
ITGAL P20701 4/20 0.49
KDM1A O60341 1/20 0.48
ALOX15 P16050 1/20 0.48
ACE P12821 4/20 0.47
MMP2 P08253 1/20 0.46
MMP9 P14780 1/20 0.46
ALDH1A1 P00352 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6551537 1.00 OPRM1 (0.50) OPRM1OPRL1ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL6727142 0.99 OPRM1 (0.49) OPRM1OPRL1ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL6727141 0.99 OPRM1 (0.49) OPRM1OPRL1ITGB2ICAM1ITGAL
SCHEMBL5164867 0.92 KMT2A (0.48) OPRM1OPRL1
Hydrochloric Acid SCHEMBL5164853 0.91 KMT2A (0.47) OPRM1OPRL1
SCHEMBL5163884 0.88 OPRL1 (0.65) OPRM1OPRL1ITGB2ICAM1ITGAL
SCHEMBL6551984 0.88 OPRL1 (0.65) OPRM1OPRL1ITGB2ICAM1ITGAL
SCHEMBL6729772 0.88 OPRL1 (0.65) OPRM1OPRL1ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL6729807 0.87 OPRL1 (0.64) OPRM1OPRL1ITGB2ICAM1ITGAL
Hydrochloric Acid SCHEMBL6729815 0.87 OPRL1 (0.64) OPRM1OPRL1ITGB2ICAM1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity GRUENENTHAL GMBH (DE) 2004-11-18 US claimed
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity GRUENENTHAL GMBH (DE) 2004-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity ARG1, CD2, PDCD1 OPRM1 250/4885OPRL1 41/4885ITGB2 2197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.