SCHEMBL5164867

SCHEMBL5164867

COC(=O)C(Cc1c[nH]c2ccccc12)NC1CCC(c2cccs2)(N(C)C)CC1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
HCRTR1 O43613 1/20 0.48
KCNA5 P22460 3/20 0.47
KCNH2 Q12809 1/20 0.47
OPRM1 P35372 3/20 0.47
OPRL1 P41146 3/20 0.47
TDP1 Q9NUW8 1/20 0.45
MAPT P10636 2/20 0.44
NPBWR1 P48145 1/20 0.44
MCHR1 Q99705 1/20 0.44
TP53 P04637 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5164853 0.99 KMT2A (0.47) KMT2AMEN1HCRTR1KCNA5KCNH2
SCHEMBL6551537 0.92 OPRM1 (0.50) OPRM1OPRL1
SCHEMBL6724438 0.92 OPRM1 (0.50) OPRM1OPRL1
Hydrochloric Acid SCHEMBL6727142 0.91 OPRM1 (0.49) OPRM1OPRL1
Hydrochloric Acid SCHEMBL6727141 0.91 OPRM1 (0.49) OPRM1OPRL1
SCHEMBL5164576 0.87 OPRL1 (0.63) KMT2AMEN1HCRTR1KCNA5KCNH2
Hydrochloric Acid SCHEMBL5165390 0.86 OPRL1 (0.62) KMT2AMEN1HCRTR1KCNA5KCNH2
SCHEMBL5164138 0.85 OPRL1 (0.52) OPRM1OPRL1
Hydrochloric Acid SCHEMBL5164593 0.84 OPRL1 (0.51) OPRM1OPRL1
SCHEMBL5858607 0.83 FPR2 (0.48) KMT2AMEN1HCRTR1KCNA5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7276518-B2 Substituted cyclohexane-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-10-02 US claimed
EP-1392641-B1 SUBSTITUTED CYCLOHEXANE-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-04-11 EP claimed
US-20040162287-A1 Substituted cyclohexane-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2004-08-19 US claimed
US-7276518-B2 Substituted cyclohexane-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2007-10-02 US disclosed
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity GRUENENTHAL GMBH (DE) 2004-11-18 US disclosed
US-20040162287-A1 Substituted cyclohexane-1,4-diamine compounds GRUENENTHAL GMBH (DE) 2004-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040162287-A1 Substituted cyclohexane-1,4-diamine compounds DPYD, DDC, QDPR KMT2A 2496/4885MEN1 1475/4885HCRTR1 1415/4885
US-20040229872-A1 Substituted cyclohexane-1,4-diamine compounds with anti-diarrhea and peripheral analgesic activity ARG1, CD2, PDCD1 KMT2A 3549/4885MEN1 4786/4885HCRTR1 1182/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.