Fumaric Acid

Fumaric Acid

SCHEMBL673089

CCCCc1nc2c(N)nc3ccccc3c2n1OCCCCN.O=C(O)/C=C/C(=O)O

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB1ADRB2ATP4AATP4BAXLCHRM2CHRM3DRD2FLT3HRH1HTR2AHTR2BHTR2CKCNH2KMT2AMAP2K1MAP2K2MEN1MLNRPLK4RENS1PR1SLC6A2SLC6A4atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 20/20 0.60
TLR8 Q9NR97 6/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Maleic Acid SCHEMBL29849281 1.00 TLR7 (0.60) TLR7TLR8
Fumaric Acid SCHEMBL673090 1.00 TLR7 (0.60) TLR7TLR8
SCHEMBL673448 0.92 TLR7 (0.69) TLR7TLR8
SCHEMBL22301797 0.87 TLR7 (0.57) TLR7TLR8
SCHEMBL18236338 0.87 TLR7 (0.60) TLR7TLR8
SCHEMBL16306624 0.86 TLR7 (0.58) TLR7TLR8
SCHEMBL19132216 0.85 TLR7 (0.63) TLR7TLR8
SCHEMBL16306619 0.85 TLR7 (0.55) TLR7TLR8
SCHEMBL23430757 0.84 TLR7 (0.56) TLR7TLR8
SCHEMBL19131056 0.84 TLR7 (0.57) TLR7TLR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12201688-B2 Lipidated immune response modifier compound compositions, formulations, and methods SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) 2025-01-21 US disclosed
US-20240252617-A1 CORONAVIRUS SPIKE PROTEIN DESIGNS, COMPOSITIONS AND METHODS FOR THEIR USE DUKE UNIVERSITY 2024-08-01 US disclosed
EP-4291569-A1 CORONAVIRUS SPIKE PROTEIN DESIGNS, COMPOSITIONS AND METHODS FOR THEIR USE Duke University (US) 2023-12-20 EP disclosed
US-20230090437-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS SOLVENTUM INTELLECTUAL PROPERTIES COMPANY 2023-03-23 US disclosed
EP-3222621-B1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND AND ITS MEDICAL USE 3M INNOVATIVE PROPERTIES COMPANY (US) 2023-03-08 EP disclosed
US-11524071-B2 Lipidated immune response modifier compound compositions, formulations, and methods 3M INNOVATIVE PROPERTIES COMPANY (US) 2022-12-13 US disclosed
WO-2022173940-A1 CORONAVIRUS SPIKE PROTEIN DESIGNS, COMPOSITIONS AND METHODS FOR THEIR USE DUKE UNIVERSITY (US) 2022-08-18 WO disclosed
US-20210038713-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS SOLVENTUM INTELLECTUAL PROPERTIES COMPANY 2021-02-11 US disclosed
US-10821176-B2 Lipidated immune response modifier compound compositions, formulations, and methods 3M INNOVATIVE PROPERTIES COMPANY (US) 2020-11-03 US disclosed
US-20200030441-A1 Lipidated Immune Response Modifier Compound Compositions, Formulations, and Methods SOLVENTUM INTELLECTUAL PROPERTIES COMPANY 2020-01-30 US disclosed
US-20170333553-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS 3M INNOVATIVE PROPERTIES CO (US) 2017-11-23 US disclosed
US-9795669-B2 Lipidated immune response modifier compound compositions, formulations, and methods 3M INNOVATIVE PROPERTIES COMPANY (US) 2017-10-24 US disclosed
EP-3222621-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND AND ITS MEDICAL USE 3M Innovative Properties Company (US) 2017-09-27 EP disclosed
US-20170189521-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS 3M INNOVATIVE PROPERTIES COMPANY (US) 2017-07-06 US disclosed
EP-2606047-B1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS 3M INNOVATIVE PROPERTIES CO (US) 2017-01-25 EP disclosed
US-20160175433-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS SOLVENTUM INTELLECTUAL PROPERTIES COMPANY 2016-06-23 US disclosed
US-9242980-B2 Lipidated immune response modifier compound compositions, formulations, and methods 3M INNOVATIVE PROPERTIES COMPANY (US) 2016-01-26 US disclosed
US-20130230578-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS 3M INNOVATIVE PROPERTIES COMPANY (US) 2013-09-05 US disclosed
EP-2606047-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS 3M Innovative Properties Company (US) 2013-06-26 EP disclosed
WO-2012024284-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS 3M INNOVATIVE PROPERTIES COMPANY (US) 2012-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10821176-B2 Lipidated immune response modifier compound compositions, formulations, and methods IFNG, MYD88, STING1 TLR7 56/4885TLR8 101/4885
US-20130230578-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS IFNG, MYD88, STING1 TLR7 56/4885TLR8 101/4885
US-20230090437-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS IRF3, IFNG, STING1 TLR7 38/4885TLR8 94/4885
US-11524071-B2 Lipidated immune response modifier compound compositions, formulations, and methods IFNG, IRF3, STING1 TLR7 79/4885TLR8 136/4885
US-20170333553-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS IFNG, MYD88, STING1 TLR7 56/4885TLR8 101/4885
US-20170189521-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS IFNG, MYD88, STING1 TLR7 56/4885TLR8 101/4885
US-20210038713-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS IFNG, IRF3, STING1 TLR7 79/4885TLR8 136/4885
US-12201688-B2 Lipidated immune response modifier compound compositions, formulations, and methods IRF3, IFNG, STING1 TLR7 38/4885TLR8 94/4885
US-20200030441-A1 Lipidated Immune Response Modifier Compound Compositions, Formulations, and Methods IFNG, MYD88, STING1 TLR7 56/4885TLR8 101/4885
US-20240252617-A1 CORONAVIRUS SPIKE PROTEIN DESIGNS, COMPOSITIONS AND METHODS FOR THEIR USE SARS1, CD14, ACE2 TLR7 2176/4885TLR8 2625/4885
US-20160175433-A1 LIPIDATED IMMUNE RESPONSE MODIFIER COMPOUND COMPOSITIONS, FORMULATIONS, AND METHODS MYD88, IFNG, STING1 TLR7 66/4885TLR8 105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.