SCHEMBL673640

SCHEMBL673640

O=C(N[C@H]1CC[C@H](C(F)(F)F)CC1)c1ccc(Cl)nc1OCC(F)F.OCC(F)F

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGES O14684 11/20 0.45
SLC6A12 P48065 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
HPGD P15428 1/20 0.37
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
IDH1 O75874 1/20 0.36
DRD2 P14416 4/20 0.36
DRD3 P35462 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL673641 1.00 PTGES (0.45) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL674097 0.97 PTGES (0.47) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL674098 0.97 PTGES (0.47) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL674115 0.84 SLC6A12 (0.39) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL674114 0.84 SLC6A12 (0.39) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL674066 0.84 SLC6A12 (0.41) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL674065 0.84 SLC6A12 (0.41) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL10091473 0.84 SLC6A12 (0.41) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL672045 0.83 CNR1 (0.42) PTGESSLC6A12CNR1CNR2HPGD
SCHEMBL672044 0.83 CNR1 (0.42) PTGESSLC6A12CNR1CNR2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2606046-A1 2-(ARYLAMINO)-3H-IMIDAZO[4,5-B]PYRIDINE-6-CARBOXAMIDE DERIVATIVES AND THEIR USE AS MPGES-1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2013-06-26 EP disclosed
WO-2012022792-A1 2-(ARYLAMINO)-3H-IMIDAZO[4,5-B]PYRIDINE-6-CARBOXAMIDE DERIVATIVES AND THEIR USE AS MPGES-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-02-23 WO disclosed