SCHEMBL6737728

SCHEMBL6737728

Nc1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 4/20 0.72
HDAC2 Q92769 2/20 0.72
HDAC8 Q9BY41 2/20 0.72
HPGD P15428 1/20 0.68
EPHX2 P34913 2/20 0.67
CA2 P00918 1/20 0.67
LMNA P02545 1/20 0.66
RAB9A P51151 1/20 0.66
HDAC1 Q13547 3/20 0.65
MAPK1 P28482 2/20 0.62
ROCK2 O75116 1/20 0.62
RPS6KA5 O75582 1/20 0.62
MAP4K4 O95819 1/20 0.62
PRKCG P05129 1/20 0.62
PRKACA P17612 1/20 0.62
RPS6KB1 P23443 1/20 0.62
AKT1 P31749 1/20 0.62
GSK3A P49840 1/20 0.62
GSK3B P49841 1/20 0.62
PRKX P51817 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3454347 0.93 HDAC6 (0.70) HDAC6HDAC2HDAC8HPGDEPHX2
SCHEMBL12604611 0.91 EPHX2 (0.78) HDAC6HDAC2HDAC8EPHX2CA2
SCHEMBL18868425 0.91 EPHX2 (0.78) HDAC6HDAC2HDAC8EPHX2CA2
SCHEMBL11900090 0.91 HDAC6 (0.85) HDAC6HDAC2HDAC8HPGDEPHX2
SCHEMBL4981515 0.90 EPHX2 (0.77) HDAC6HDAC2HDAC8EPHX2CA2
Hydrochloric Acid SCHEMBL30918901 0.89 EPHX2 (0.76) HDAC6HDAC2HDAC8EPHX2CA2
Succinic Acid SCHEMBL11587387 0.87 HDAC1 (0.62) HDAC6HDAC2HDAC8HPGDEPHX2
SCHEMBL457082 0.87 HDAC6 (0.79) HDAC6HDAC2HDAC8HPGDEPHX2
SCHEMBL6140514 0.86 HDAC6 (0.72) HDAC6HDAC2HDAC8HPGDEPHX2
SCHEMBL6843720 0.85 HDAC6 (0.77) HDAC6HDAC2HDAC8HPGDEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 55 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025085689-A1 EXTRACELLULAR SMALL MOLECULE ACTIVATORS TARGETING BESTROPHIN CHANNELS FOR DISEASE TREATMENT THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2025-04-24 WO claimed
EP-0078845-B1 ANTI-CONVULSANT CLARK, Charles Randall (US) 1987-02-04 EP claimed
EP-0078845-A4 ANTI-CONVULSANT. CLARK CHARLES RANDALL 1983-09-02 EP claimed
EP-0078845-A1 ANTI-CONVULSANT. CLARK CHARLES RANDALL 1983-05-18 EP claimed
US-4379165-A Anti-convulsant RESEARCH CORPORATION (US) 1983-04-05 US claimed
WO-1982004046-A1 ANTI-CONVULSANT CLARK CHARLES RANDALL 1982-11-25 WO claimed
WO-2025085689-A1 EXTRACELLULAR SMALL MOLECULE ACTIVATORS TARGETING BESTROPHIN CHANNELS FOR DISEASE TREATMENT THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2025-04-24 WO disclosed
US-10752624-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2020-08-25 US disclosed
US-20180305356-A1 NOVEL KINASE INHIBITORS ORIGENIS GMBH (DE) 2018-10-25 US disclosed
US-10000482-B2 Kinase inhibitors ORIGENIS GMBH (DE) 2018-06-19 US disclosed
US-9637491-B2 Pyrazolo[4,3-D]pyrimidines as kinase inhibitors ORIGENIS GMBH (DE) 2017-05-02 US disclosed
CN-104478780-B Acylpyrrole small-molecular organic compound, derivatives of organic compound as well as application and preparation method of acylpyrrole small-molecular organic compound and derivatives of organic compound 华东师范大学 2017-04-19 CN disclosed
EP-2488032-B1 PROSTAGLANDIN TRANSPORTER INHIBITORS AND USES THEREOF EINSTEIN COLL MED (US) 2016-11-02 EP disclosed
EP-0078845-A4 ANTI-CONVULSANT. CLARK CHARLES RANDALL 1983-09-02 EP disclosed
EP-0078845-A1 ANTI-CONVULSANT. CLARK CHARLES RANDALL 1983-05-18 EP disclosed
US-4379165-A Anti-convulsant RESEARCH CORPORATION (US) 1983-04-05 US disclosed
WO-1982004046-A1 ANTI-CONVULSANT CLARK CHARLES RANDALL 1982-11-25 WO disclosed
US-4118503-A ANTIULCER AGENTS PFIZER INC. (US) 1978-10-03 US disclosed
US-4117138-A ANTIULCER PFIZER INC. (US) 1978-09-26 US disclosed
US-4064264-A Pyrrolidonecarboxylic acid derivatives as anti-ulcer agents PFIZER INC. (US) 1977-12-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180305356-A1 NOVEL KINASE INHIBITORS LRRK2, MYLK2, MYLK HDAC6 1604/4885HDAC2 1409/4885HDAC8 3493/4885
US-10000482-B2 Kinase inhibitors LRRK2, MYLK2, MYLK HDAC6 1677/4885HDAC2 1530/4885HDAC8 3648/4885
US-10752624-B2 Kinase inhibitors LRRK2, MYLK2, MYLK HDAC6 1677/4885HDAC2 1530/4885HDAC8 3648/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.