SCHEMBL6739701

SCHEMBL6739701

COC(=O)C(O)=CC(=O)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 1/20 0.32
TET2 Q6N021 1/20 0.31
EGLN1 Q9GZT9 1/20 0.31
HCAR2 Q8TDS4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6739700 1.00 MAPK1 (0.37) MAPK1RAB9AHSD17B10NPC1TSHR
SCHEMBL10116679 0.83 ALDH1A1 (0.30) ALDH1A1KDM4EMAPT
SCHEMBL3576290 0.77 NPSR1 (0.44) MAPK1RAB9AHSD17B10NPC1TSHR
SCHEMBL3576293 0.77 NPSR1 (0.44) MAPK1RAB9AHSD17B10NPC1TSHR
SCHEMBL10175722 0.76 MAPK1 (0.39) MAPK1RAB9AHSD17B10NPC1TSHR
SCHEMBL27714278 0.75 HCAR2 (0.40) TSHRALDH1A1KDM4EMAPTTET2
SCHEMBL15563291 0.75 TSHR (0.37) MAPK1RAB9AHSD17B10NPC1TSHR
SCHEMBL15563292 0.75 TSHR (0.37) MAPK1RAB9AHSD17B10NPC1TSHR
SCHEMBL15873736 0.74 DGAT1 (0.39) ALDH1A1KDM4EMAPTHCAR2
SCHEMBL12348409 0.73 ALDH1A1 (0.42) ALDH1A1KDM4EMAPTTET2EGLN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6713503-B1 1-(2,4-DIMETHYL-PHENYL)-2,4-DIHYDROXY-3-(4-METHYL-BENZOYL)-5-OXO-2,5 -DIHYDRO-1H-PYRROLE-2-CARBOXYLIC ACID METHYL ESTER UNIVERSITY OF CENTRAL FLORIDA 2004-03-30 US disclosed
US-6703426-B1 4-(4-CHLORO-PHENYL)-2,4-DIOXO-3- (PHENYL-HYDRAZONO)-BUTYRIC ACID ETHYL ESTER IS ADMINISTERED UNIVERSITY OF CENTRAL FLORIDA 2004-03-09 US disclosed
US-6686496-B1 4-OXO-2 BUTENOIC ACID AND 3-HYDRAZINO-2,4-DIOXOBUTANOIC ACID DERIVATIVES UNIVERSITY OF CENTRAL FLORIDA 2004-02-03 US disclosed
US-6683110-B1 4-(4-ETHOXYPHENYL)-2-(N'-FLUOREN-9-YLIDENEHYDRAZINO)-2-HYDROXY -4-OXOBUTYRIC ACID METHYL ESTER; 2-(4-BROMOPHENYL-AMINO)-5,5-DIMETHYL-4-OXOHEX-2-ENOIC ACID METHYL ESTER UNIVERSITY OF CENTRAL FLORIDA 2004-01-27 US disclosed
US-6638975-B1 Treatment of breast cancer UNIVERSITY OF CENTRAL FLORIDA 2003-10-28 US disclosed
US-6602907-B1 Treatment of breast cancer UNIVERSITY OF CENTRAL FLORIDA 2003-08-05 US disclosed