SCHEMBL6742547

SCHEMBL6742547

[CH2]Cc1cc(C)cc(NC=O)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
TACR1 P25103 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31
HDAC5 Q9UQL6 1/20 0.31
THRB P10828 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL424461 0.80 ALDH1A1 (0.44) ALDH1A1HTTNPSR1KDM4ECYP1A2
SCHEMBL1706527 0.72 ALDH1A1 (0.40) ALDH1A1TACR1HTTNPSR1
SCHEMBL17748457 0.71 RAPGEF4 (0.42) ALDH1A1KDM4EHDAC3HDAC1HDAC2
SCHEMBL6740662 0.70 NPSR1 (0.34) ALDH1A1NPSR1KDM4ECYP3A4
SCHEMBL838486 0.70 ALDH1A1 (0.50) ALDH1A1THRBLMNA
SCHEMBL7380802 0.69 MAPT (0.44) ALDH1A1HTTNPSR1KDM4ECYP1A2
SCHEMBL6740663 0.68 ALDH1A1 (0.39) ALDH1A1HTTNPSR1CYP1A2CYP3A4
SCHEMBL1588979 0.67 ALDH1A1 (0.55) ALDH1A1LMNA
SCHEMBL18257145 0.67 SAE1 (0.45) ALDH1A1HTTKDM4ECYP1A2CYP3A4
SCHEMBL7352511 0.66 ALDH1A1 (0.44) ALDH1A1NPC1LMNARAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6689771-B2 TREATMENT OF RHEUMATOID ARTHRITIS, OSTEOARTHRITIS, PERIODONTITIS, GINGIVITIS, CORNEAL ULCERATION, SOLID TUMOR GROWTH BRISTOL-MYERS SQUIBB PHARMA COMPANY 2004-02-10 US disclosed
US-6376665-B1 ANTIARTHRITIC AGENTS, ANTIINFLAMMATORY AGENTS BRISTOL-MYERS SQUIBB PHARMA COMPANY 2002-04-23 US disclosed