Aniline

Aniline

SCHEMBL675043

Nc1ccccc1.Nc1ccccc1.Nc1ccccc1.O=P(O)(O)O

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Aniline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.65
CA2 P00918 1/20 0.50
CA4 P22748 1/20 0.50
CA5A P35218 1/20 0.50
PBRM1 Q86U86 1/20 0.48
CYP3A4 P08684 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
HSD17B10 Q99714 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
SRC P12931 2/20 0.44
CFTR P13569 1/20 0.44
FDPS P14324 3/20 0.43
PTPN1 P18031 1/20 0.42
LAP3 P28838 3/20 0.41
ANPEP P15144 1/20 0.41
ALOX15 P16050 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aniline SCHEMBL5334646 1.00 TSHR (0.65) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL321169 1.00 TSHR (0.65) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL29573098 1.00 TSHR (0.65) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL28659856 0.97 TSHR (0.61) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL1533980 0.97 TSHR (0.61) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL28661396 0.97 TSHR (0.61) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL28663674 0.97 TSHR (0.61) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL8683062 0.92 TSHR (0.61) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL6538352 0.90 TSHR (0.52) TSHRCA2CA4CA5APBRM1
Aniline SCHEMBL28527754 0.90 TSHR (0.52) TSHRCA2CA4CA5APBRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116323817-A Powder composition, coating film and three-dimensional molded article 大金工业株式会社 2023-06-23 CN disclosed
CN-113563138-A Method for reducing soil nitrogen emission and nitrogen emission inhibitor used by same 浙江省农业科学院 2021-10-29 CN disclosed
CN-104854224-B Lubricating grease composition for improving low-temperature fretting 协同油脂株式会社 2020-03-24 CN disclosed
EP-2920148-B1 PICTET-SPENGLER LIGATION FOR PROTEIN CHEMICAL MODIFICATION UNIV CALIFORNIA (US) 2019-06-12 EP disclosed
US-9605078-B2 Pictet-Spengler ligation for protein chemical modification THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-03-28 US disclosed
US-20150291699-A1 PICTET-SPENGLER LIGATION FOR PROTEIN CHEMICAL MODIFICATION GERAWAN FARMING LLC 2015-10-15 US disclosed
EP-2920148-A1 PICTET-SPENGLER LIGATION FOR PROTEIN CHEMICAL MODIFICATION The Regents of The University of California (US) 2015-09-23 EP disclosed
WO-2014078733-A1 PICTET-SPENGLER LIGATION FOR PROTEIN CHEMICAL MODIFICATION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2014-05-22 WO disclosed
US-7968009-B2 Electrically conductive nanocomposite particles having a polyalkyl acrylate core and a polyaniline coating UPPA-UNIVERSITE DE PAU ET DES PAYS DE L'ADOUR (FR) 2011-06-28 US disclosed
US-20090212263-A1 ELECTRICALLY CONDUCTIVE NANOCOMPOSITE PARTICLES HAVING A POLYALKYL ACRYLATE CORE AND A POLYANILINE COATING CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2009-08-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150291699-A1 PICTET-SPENGLER LIGATION FOR PROTEIN CHEMICAL MODIFICATION PTMS, SHMT1, OGA TSHR 1153/4885CA2 1936/4885CA4 890/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.